SCHEMBL572754

SCHEMBL572754

CC(C)(C)OC(=O)NCC(C(=O)NC(CC(=O)N1CCCC1C(N)=O)Cc1cc(F)c(F)cc1F)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.44
DPP4 P27487 17/20 0.42
DPP8 Q6V1X1 15/20 0.42
DPP9 Q86TI2 15/20 0.42
DPP7 Q9UHL4 15/20 0.42
CYP2D6 P10635 8/20 0.42
ACE P12821 1/20 0.41
ELANE P08246 1/20 0.38
PREP P48147 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10057885 0.85 ACE (0.55) KLK5ACE
SCHEMBL572136 0.85 ACE (0.55) KLK5ACE
SCHEMBL10056843 0.79 ACE (0.48) DPP4DPP8DPP9DPP7CYP2D6
Trifluoroacetic Acid SCHEMBL572058 0.77 DPP4 (0.47) DPP4DPP8DPP9DPP7CYP2D6
SCHEMBL10057504 0.77 ACE (0.51) KLK5DPP4DPP8DPP9DPP7
SCHEMBL572693 0.73 ACE (0.49) KLK5DPP4DPP8ACEPREP
SCHEMBL14982904 0.73 ACE (0.49) KLK5DPP4DPP8ACEPREP
SCHEMBL6693358 0.72 KLK5 (0.54) KLK5DPP4ACEELANE
SCHEMBL6693361 0.72 KLK5 (0.54) KLK5DPP4ACEELANE
SCHEMBL14102471 0.71 KLK5 (0.54) KLK5DPP4DPP9ACEPREP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2600888-A2 NOVEL COMPOUNDS AS DPP-IV INHIBITORS AND PROCESS FOR PREPARATION THEREOF Cadila Pharmaceuticals Ltd. (IN) 2013-06-12 EP disclosed
WO-2012017391-A2 NOVEL COMPOUNDS AS DPP-IV INHIBITORS AND PROCESS FOR PREPARATION THEREOF CADILA PHARMACEUTICALS LIMITED (IN) 2012-02-09 WO disclosed