SCHEMBL5728078

SCHEMBL5728078

C[C@H]1CC[C@H](C(=O)N(c2sc(-c3ccccc3)cc2OC(=O)O)C2CCNCC2)CC1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
HTT P42858 1/20 0.36
ATM Q13315 1/20 0.36
CHEK1 O14757 3/20 0.36
SLC6A2 P23975 12/20 0.35
SLC6A4 P31645 12/20 0.35
CHRM1 P11229 1/20 0.35
SLC6A3 Q01959 9/20 0.34
KCNH2 Q12809 7/20 0.34
CYP2D6 P10635 4/20 0.34
CHRM3 P20309 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5728684 0.91 SLC6A2 (0.38) KDM4ECHEK1SLC6A2SLC6A4CHRM1
SCHEMBL5728123 0.88 KDM4E (0.36) KDM4EHTTATMCHEK1
SCHEMBL5433037 0.86 CHEK1 (0.41) KDM4EHTTATMCHEK1SLC6A2
SCHEMBL5433041 0.86 CHEK1 (0.41) KDM4EHTTATMCHEK1SLC6A2
SCHEMBL5438394 0.85 ALDH1A1 (0.45) KDM4EHTTATMCHEK1SLC6A2
SCHEMBL5438391 0.85 ALDH1A1 (0.45) KDM4EHTTATMCHEK1SLC6A2
SCHEMBL2871147 0.85 KDM4E (0.36) KDM4EHTTATMCHEK1SLC6A2
SCHEMBL5728035 0.85 OPRM1 (0.35) KDM4EHTTATMCHRM3
SCHEMBL5430676 0.84 ALDH1A1 (0.48) KDM4EHTTSLC6A2SLC6A4SLC6A3
SCHEMBL5430668 0.84 ALDH1A1 (0.48) KDM4EHTTSLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694665-A2 SUBSTITUTED THIOPHENES AiCuris GmbH & Co. KG (DE) 2006-08-30 EP disclosed
WO-2005063734-A2 SUBSTITUTED THIOPHENES AICURIS GMBH & CO. KG (DE) 2005-07-14 WO disclosed