SCHEMBL5728540

SCHEMBL5728540

CC(=O)C(C)(C)Cc1ccc(CBr)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
BLM P54132 2/20 0.38
ESR1 P03372 3/20 0.38
THRA P10827 1/20 0.37
THRB P10828 1/20 0.37
KMT2A Q03164 3/20 0.36
TSHR P16473 2/20 0.36
MEN1 O00255 2/20 0.36
ALDH1A1 P00352 4/20 0.35
TRPA1 O75762 1/20 0.34
ESR2 Q92731 2/20 0.34
GRN P28799 1/20 0.34
SORT1 Q99523 1/20 0.34
CYP4F2 P78329 1/20 0.33
CYP4A11 Q02928 1/20 0.33
CYP3A4 P08684 3/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5728742 0.85 MEN1 (0.47) BLMESR1THRATHRBKMT2A
SCHEMBL10767808 0.84 LMNA (0.42) BLMESR1THRATHRBKMT2A
SCHEMBL8951998 0.82 HPGD (0.44) CES2CES1BLMESR1THRA
SCHEMBL9626513 0.80 RIPK1 (0.47) BLMKMT2AMEN1TRPA1KDM4E
SCHEMBL2442200 0.80 EPHX2 (0.47) KMT2AMEN1CYP1A2CYP2C19LMNA
SCHEMBL10383881 0.80 SLC6A4 (0.53) KMT2AMEN1ALDH1A1GRNSORT1
SCHEMBL5567033 0.79 PTPRB (0.42) CES2CES1BLMKMT2ATSHR
SCHEMBL6552350 0.79 SMN1; SMN2 (0.50) ALDH1A1TRPA1CYP3A4CYP1A2CYP2D6
SCHEMBL5729103 0.78 PPARA (0.49) BLMESR1THRATHRBTSHR
Ammonia Solution, Strong SCHEMBL11617477 0.78 SMN1; SMN2 (0.48) ALDH1A1TRPA1CYP3A4CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720836-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO [D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2006-11-15 EP disclosed
WO-2005082859-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2005-09-09 WO disclosed