SCHEMBL5728826

SCHEMBL5728826

[CH2]C(OS(C)(=O)=O)c1nccs1

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.32
MAPKAPK2 P49137 1/20 0.31
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL507287 0.81 ALDH1A1 (0.35) ALDH1A1MAPKAPK2PKM
SCHEMBL8427577 0.70 ALDH1A1 (0.34) ALDH1A1MAPKAPK2PKM
SCHEMBL2838919 0.69 ALDH1A1 (0.34) ALDH1A1MAPKAPK2
SCHEMBL1987440 0.69
SCHEMBL17530037 0.67 MAPKAPK2 (0.43) ALDH1A1MAPKAPK2
SCHEMBL2949467 0.66 ALDH1A1 (0.40) ALDH1A1PKM
SCHEMBL7804726 0.65
SCHEMBL4137927 0.65
SCHEMBL28842884 0.65
SCHEMBL8267529 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720836-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO [D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2006-11-15 EP disclosed
WO-2005082859-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2005-09-09 WO disclosed