SCHEMBL573254

SCHEMBL573254

O=C(CCCCCCNC(=O)c1ccccc1)NO

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 17/20 1.00
HDAC1 Q13547 12/20 1.00
HDAC8 Q9BY41 12/20 1.00
HDAC3 O15379 10/20 1.00
HDAC4 P56524 10/20 1.00
HDAC2 Q92769 10/20 1.00
HDAC10 Q969S8 10/20 1.00
HDAC11 Q96DB2 10/20 1.00
HDAC9 Q9UKV0 10/20 1.00
HDAC5 Q9UQL6 10/20 1.00
HDAC7 Q8WUI4 9/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1232912 1.00 HDAC6 (1.00) HDAC6HDAC1HDAC8HDAC3HDAC4
SCHEMBL1232629 0.98 HDAC6 (0.97) HDAC6HDAC1HDAC8HDAC3HDAC4
SCHEMBL6386847 0.93 HDAC6 (0.88) HDAC6HDAC1HDAC8HDAC3HDAC4
Trifluoroacetic Acid SCHEMBL29825044 0.92 HDAC6 (0.84) HDAC6HDAC1HDAC8HDAC3HDAC4
SCHEMBL6387051 0.91 HDAC6 (1.00) HDAC6HDAC1HDAC8HDAC3HDAC4
SCHEMBL6385727 0.91 HDAC6 (1.00) HDAC6HDAC1HDAC8HDAC3HDAC4
SCHEMBL6389005 0.89 HDAC6 (0.97) HDAC6HDAC1HDAC8HDAC3HDAC4
SCHEMBL2226579 0.89 HDAC6 (1.00) HDAC6HDAC1HDAC8HDAC3HDAC4
SCHEMBL4922807 0.88 HDAC1 (1.00) HDAC6HDAC1HDAC8HDAC3HDAC4
SCHEMBL4258321 0.88 HDAC1 (1.00) HDAC6HDAC1HDAC8HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3455204-B1 CYCLOPROPYL-AMIDE COMPOUNDS AS DUAL LSD1/HDAC INHIBITORS Jubilant Epicore LLC (US) 2025-10-29 EP claimed
US-20050119305-A1 Il-6 production inhibitors ONO PHARMACEUTICAL CO., LTD. (JP) 2005-06-02 US claimed
CN-115141123-B Compound, preparation method thereof and application thereof in preparation of dual inhibitors of histone deacetylase and epoxide hydrolase 沈阳药科大学 2024-05-17 CN disclosed
CN-117843548-A Benzyl indole HDAC inhibitor and pharmaceutical application thereof 南京医科大学 2024-04-09 CN disclosed
CN-115141123-A Compound, preparation method thereof and application thereof in preparation of histone deacetylase and epoxide hydrolase dual inhibitor 沈阳药科大学 2022-10-04 CN disclosed
EP-2839037-B1 BIOMARKERS TO IDENTIFY PATIENTS THAT WILL RESPOND TO TREATMENT AND TREATING SUCH PATIENTS ACETYLON PHARMACEUTICALS INC (US) 2018-12-26 EP disclosed
WO-2017133517-A1 PHOSPHAMIDE DERIVATIVE, METHOD FOR MANUFACTURING THE SAME, AND USES THEREOF 四川海思科制药有限公司 2017-08-10 WO disclosed
US-8394810-B2 Reverse amide compounds as protein deacetylase inhibitors and methods of use thereof ACETYLON PHARMACEUTICALS (US) 2013-03-12 US disclosed
US-20110300134-A1 REVERSE AMIDE COMPOUNDS AS PROTEIN DEACETYLASE INHIBITORS AND METHODS OF USE THEREOF ACETYLON PHARMACEUTICALS (US) 2011-12-08 US disclosed
EP-1443928-B1 TREATMENT OF NEURODEGENERATIVE DISEASES AND CANCER OF THE BRAIN SLOAN KETTERING INST CANCER (US) 2011-07-27 EP disclosed
US-20050119305-A1 Il-6 production inhibitors ONO PHARMACEUTICAL CO., LTD. (JP) 2005-06-02 US disclosed
WO-2003032921-A2 TREATMENT OF NEURODEGENERATIVE DISEASES AND CANCER OF THE BRAIN SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2003-04-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110300134-A1 REVERSE AMIDE COMPOUNDS AS PROTEIN DEACETYLASE INHIBITORS AND METHODS OF USE THEREOF HDAC6, HDAC1, HDAC3 HDAC6 1/4885HDAC1 2/4885HDAC8 6/4885
US-20050119305-A1 Il-6 production inhibitors IL6, IL6ST, PADI6 HDAC6 2866/4885HDAC1 1343/4885HDAC8 1593/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.