SCHEMBL5733440

SCHEMBL5733440

COC(=O)Oc1ccc2nc(Nc3ccc(Oc4ccncc4)cc3)[nH]c2c1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.56
RAF1 P04049 10/20 0.56
BRAF P15056 9/20 0.56
TEK Q02763 3/20 0.51
CSNK1A1 P48729 1/20 0.50
CSNK1D P48730 1/20 0.50
ALDH1A1 P00352 1/20 0.49
HPGD P15428 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5733146 0.89 KDR (0.58) KDRRAF1BRAFTEKCSNK1A1
SCHEMBL4173612 0.85 RAF1 (0.55) KDRRAF1BRAFTEKCSNK1A1
SCHEMBL4166869 0.82 POLB (0.61) KDRRAF1BRAFTEKCSNK1A1
SCHEMBL5734205 0.82 RAF1 (0.41) KDRRAF1BRAFTEKCSNK1A1
SCHEMBL4158747 0.82 KDR (0.59) KDRRAF1BRAFCSNK1A1CSNK1D
SCHEMBL13906245 0.79 KDR (0.59) KDRRAF1BRAFTEKCSNK1A1
SCHEMBL13906239 0.79 KDR (0.54) KDRRAF1BRAFTEKCSNK1A1
SCHEMBL4164763 0.78 KDR (0.54) KDRRAF1BRAFTEKCSNK1A1
SCHEMBL4161824 0.77 CSNK1D (0.80) KDRRAF1BRAFCSNK1A1CSNK1D
SCHEMBL4164501 0.77 RIPK1 (0.67) KDRRAF1BRAFCSNK1A1CSNK1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1675849-A1 BENZIMIDAZOLYL DERIVATIVES MERCK PATENT GmbH (DE) 2006-07-05 EP claimed
WO-2005042520-A1 BENZIMIDAZOLYL DERIVATIVES MERCK PATENT GMBH (DE) 2005-05-12 WO claimed
EP-1675849-A1 BENZIMIDAZOLYL DERIVATIVES MERCK PATENT GmbH (DE) 2006-07-05 EP disclosed
WO-2005042520-A1 BENZIMIDAZOLYL DERIVATIVES MERCK PATENT GMBH (DE) 2005-05-12 WO disclosed