SCHEMBL5733657

SCHEMBL5733657

NC(=O)c1ccc2ccn(N3CCC(Cc4ccccc4)CC3)c2c1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.55
F2 P00734 2/20 0.50
ACHE P22303 1/20 0.49
TNKS O95271 1/20 0.46
PARP1 P09874 1/20 0.46
PARP14 Q460N5 1/20 0.46
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5203573 0.91 F2 (0.57) GAAF2ACHETNKSPARP1
SCHEMBL5374204 0.82 CYP2C9 (0.47) GAAF2MEN1KMT2A
SCHEMBL5374688 0.81 GAA (0.47) GAAF2ACHE
SCHEMBL5733306 0.80 ROCK2 (0.51) GAAF2ACHETNKSPARP1
SCHEMBL5201672 0.79 MEN1 (0.57) F2ACHEMEN1KMT2A
SCHEMBL5372863 0.78 F2 (0.59) GAAF2TNKSPARP1PARP14
SCHEMBL5734925 0.77 F2 (0.47) GAAF2ACHE
SCHEMBL7376188 0.76 GAA (0.53) GAAF2ACHETNKSPARP1
SCHEMBL5377979 0.76 GAA (0.47) GAAF2ACHETNKSPARP1
SCHEMBL5732645 0.75 F2 (0.50) GAAF2ACHETNKSPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1080078-B1 HETEROCYCLIC COMPOUNDS AND METHODS TO TREAT CARDIAC FAILURE AND OTHER DISORDERS SCIOS INC (US) 2006-02-01 EP disclosed
US-6589954-B1 Indoles, benzimidazoles and benztriazoles which are substituted at the 5 or 6 position with a substituent comprising an aromatic moiety linked through a piperazine ring to said indole, benzimidazole or benztriazole are useful SCIOS, INC. 2003-07-08 US disclosed