SCHEMBL5732645

SCHEMBL5732645

NC(=O)c1ccc2c(ccn2N2CCC(Cc3ccccc3)CC2Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F2 P00734 4/20 0.50
GAA P10253 1/20 0.49
OPRM1 P35372 1/20 0.44
OPRD1 P41143 1/20 0.44
OPRK1 P41145 1/20 0.44
KCNH2 Q12809 1/20 0.44
ACHE P22303 2/20 0.42
TNKS O95271 1/20 0.40
PARP1 P09874 1/20 0.40
PARP14 Q460N5 1/20 0.40
HDAC6 Q9UBN7 1/20 0.39
MGLL Q99685 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5374213 0.88 F2 (0.50) F2GAAOPRM1OPRD1OPRK1
SCHEMBL5203573 0.83 F2 (0.57) F2GAAACHETNKSPARP1
SCHEMBL5374688 0.76 GAA (0.47) F2GAAACHEHDAC6
SCHEMBL5733306 0.75 ROCK2 (0.51) F2GAAOPRM1OPRD1OPRK1
SCHEMBL5733657 0.75 GAA (0.55) F2GAAACHETNKSPARP1
SCHEMBL5732647 0.74 GAA (0.48) GAAOPRM1OPRD1OPRK1KCNH2
SCHEMBL7076353 0.73 PARP14 (0.39) F2OPRM1OPRD1PARP14
SCHEMBL5734925 0.72 F2 (0.47) F2GAAACHE
SCHEMBL5733400 0.71 ROCK2 (0.41) F2GAAOPRM1OPRD1OPRK1
SCHEMBL5371447 0.69 HDAC6 (0.55) F2GAAACHETNKSPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1080078-B1 HETEROCYCLIC COMPOUNDS AND METHODS TO TREAT CARDIAC FAILURE AND OTHER DISORDERS SCIOS INC (US) 2006-02-01 EP claimed