SCHEMBL5735196

SCHEMBL5735196

NC(=O)c1cc2ccc(Cl)cc2n1N1CCC(Cc2ccc(F)cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GMNN O75496 1/20 0.43
TP53 P04637 1/20 0.43
CYP3A4 P08684 1/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43
THPO P40225 1/20 0.43
MTOR P42345 1/20 0.43
BLM P54132 1/20 0.43
GRIN1 Q05586 1/20 0.43
GRIN2B Q13224 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
RPS6KB1 P23443 1/20 0.39
GAA P10253 1/20 0.39
PLA2G10 O15496 1/20 0.38
PLA2G2A P14555 1/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
CCR3 P51677 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7078849 0.77 GAA (0.49) GAAPLA2G10
SCHEMBL5376287 0.73 MAPK14 (0.43) GMNNTP53CYP3A4ALOX15TSHR
SCHEMBL5374688 0.69 GAA (0.47) GAA
SCHEMBL5806708 0.68 MEN1 (0.55) GRIN1GRIN2BCCR3
SCHEMBL5387256 0.68 ALOX15 (0.42) GMNNTP53CYP3A4ALOX15TSHR
SCHEMBL5378327 0.67 CCR3 (0.40) GMNNTP53CYP3A4ALOX15TSHR
Hydrochloric Acid SCHEMBL27943768 0.67 MEN1 (0.54) CCR3
SCHEMBL5732819 0.67 MEN1 (0.46) CCR3
SCHEMBL21614171 0.66 MEN1 (0.53) GRIN1GRIN2BCCR3
SCHEMBL14439429 0.66 GRIN2B (0.52) GMNNTP53CYP3A4ALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1080078-B1 HETEROCYCLIC COMPOUNDS AND METHODS TO TREAT CARDIAC FAILURE AND OTHER DISORDERS SCIOS INC (US) 2006-02-01 EP claimed