SCHEMBL5738475

SCHEMBL5738475

O=CC(Br)c1ccc(Oc2cccc([N+](=O)[O-])c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
LTA4H P09960 1/20 0.47
PTGS2 P35354 1/20 0.47
KDM4E B2RXH2 1/20 0.46
NPY5R Q15761 1/20 0.44
PGR P06401 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
LPAR3 Q9UBY5 1/20 0.43
LMNA P02545 3/20 0.42
MEN1 O00255 2/20 0.42
MAPT P10636 2/20 0.42
KMT2A Q03164 2/20 0.42
TSHR P16473 1/20 0.42
NFE2L2 Q16236 1/20 0.40
FFAR1 O14842 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNA4 P43681 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL40530 0.86 HSPB1 (0.53) ALDH1A1LTA4HPTGS2KDM4ELMNA
SCHEMBL9158141 0.82 ALDH1A1 (0.67) ALDH1A1LTA4HPTGS2KDM4EPGR
SCHEMBL9356592 0.82 ALDH1A1 (0.67) ALDH1A1LTA4HPTGS2KDM4EPGR
SCHEMBL15472357 0.80 ALDH1A1 (0.54) ALDH1A1LTA4HPTGS2KDM4ENPY5R
SCHEMBL1701431 0.79 TSHR (0.53) ALDH1A1LMNAMEN1MAPTKMT2A
SCHEMBL9214229 0.79 ALDH1A1 (0.73) ALDH1A1LTA4HPTGS2KDM4EPGR
SCHEMBL4203388 0.79 TSHR (0.67) ALDH1A1LTA4HPTGS2KDM4ECYP2C9
SCHEMBL9687087 0.78 ALDH1A1 (0.58) ALDH1A1LTA4HPTGS2KDM4ENPY5R
SCHEMBL8775401 0.78 ALDH1A1 (0.61) ALDH1A1LTA4HPTGS2KDM4EPGR
SCHEMBL30042572 0.78 ALDH1A1 (0.61) ALDH1A1LTA4HPTGS2KDM4EPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1638943-A2 NOVEL IMIDAZOLE DERIVATIVES, THE PRODUCTION THEREOF, AND THE USE OF THE SAME AS A MEDICAMENT Société de Conseils de Recherches et d'Applications Scientifiques ( S.C.R.A.S.) (FR) 2006-03-29 EP disclosed
WO-2004106307-A2 NOVEL IMIDAZOLE DERIVATIVES, THE PRODUCTION THEREOF, AND THE USE OF THE SAME AS A MEDICAMENT SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2004-12-09 WO disclosed