SCHEMBL5739062

SCHEMBL5739062

CCCCNc1ncnn2cc(OC(=O)OCC)c(CC)c12

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EGFR P00533 8/20 0.49
ERBB2 P04626 8/20 0.49
KDR P35968 3/20 0.42
MAPK14 Q16539 6/20 0.38
MAP2K1 Q02750 1/20 0.36
MAP4K4 O95819 1/20 0.35
PDE5A O76074 1/20 0.35
PDE4B Q07343 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5740220 0.89 EGFR (0.48) EGFRERBB2KDRMAPK14
SCHEMBL5741109 0.85 EGFR (0.45) EGFRERBB2
SCHEMBL5739083 0.85 EGFR (0.59) EGFRERBB2KDRMAP2K1
SCHEMBL5512127 0.83 EGFR (0.70) EGFRERBB2KDRMAPK14MAP2K1
SCHEMBL5740547 0.83 EGFR (0.50) EGFRERBB2KDRMAPK14MAP2K1
SCHEMBL5739637 0.83 EGFR (0.72) EGFRERBB2MAPK14MAP2K1
SCHEMBL5739177 0.81 EGFR (0.46) EGFRERBB2KDRMAPK14MAP2K1
SCHEMBL5741061 0.81 EGFR (0.46) EGFRERBB2KDRMAPK14MAP2K1
SCHEMBL5740236 0.81 EGFR (0.59) EGFRERBB2KDRMAPK14MAP2K1
SCHEMBL5740085 0.80 EGFR (0.62) EGFRERBB2KDRMAPK14MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183033-B1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL MYERS SQUIBB CO (US) 2006-03-01 EP claimed