SCHEMBL5740236

SCHEMBL5740236

CCOC(=O)Oc1cn2ncnc(NCc3ccc(Br)cc3)c2c1CC

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.59
ERBB2 P04626 7/20 0.59
KDR P35968 3/20 0.37
GAA P10253 1/20 0.37
AURKA O14965 1/20 0.36
RPS6KB1 P23443 1/20 0.36
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
GLA P06280 1/20 0.35
MAP2K1 Q02750 1/20 0.35
MAPK14 Q16539 3/20 0.35
MAP4K4 O95819 1/20 0.34
KIT P10721 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5739637 0.90 EGFR (0.72) EGFRERBB2GAAALDH1A1LMNA
SCHEMBL5742139 0.89 EGFR (0.58) EGFRERBB2KDRAURKARPS6KB1
SCHEMBL5739277 0.87 EGFR (0.58) EGFRERBB2KDRMAP2K1MAPK14
SCHEMBL4044139 0.85 EGFR (0.82) EGFRERBB2KDRGAAMAP2K1
SCHEMBL5739062 0.81 EGFR (0.49) EGFRERBB2KDRMAP2K1MAPK14
SCHEMBL5739083 0.81 EGFR (0.59) EGFRERBB2KDRALDH1A1LMNA
SCHEMBL5740220 0.81 EGFR (0.48) EGFRERBB2KDRALDH1A1MAPK14
SCHEMBL5740575 0.80 EGFR (0.74) EGFRERBB2KDRMAP2K1
SCHEMBL5740085 0.79 EGFR (0.62) EGFRERBB2KDRMAP2K1MAPK14
SCHEMBL5740274 0.78 EGFR (0.56) EGFRERBB2KDRMAP2K1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183033-B1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL MYERS SQUIBB CO (US) 2006-03-01 EP claimed