SCHEMBL5740250

SCHEMBL5740250

COc1ccc2nccc(-c3ccc(CC(NC(=O)O)C(C)(C)C)nc3)c2n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.35
SLC22A12 Q96S37 1/20 0.34
PIK3CG P48736 2/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
WNT3A P56704 1/20 0.33
F9 P00740 1/20 0.33
F10 P00742 1/20 0.33
F11 P03951 1/20 0.33
PRSS1 P07477 1/20 0.33
PRSS2 P07478 1/20 0.33
F7 P08709 1/20 0.33
PRSS3 P35030 1/20 0.33
AAK1 Q2M2I8 2/20 0.33
PDE10A Q9Y233 1/20 0.32
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
OXTR P30559 1/20 0.32
SLC2A1 P11166 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2917178 0.79 MTNR1A (0.40) KCNH2PIK3CGPIK3CDPIK3CAPIK3CB
SCHEMBL13175635 0.77 MTNR1A (0.40) KCNH2AAK1
SCHEMBL13175669 0.74 RPS6KA3 (0.36) KCNH2PIK3CGPIK3CDPIK3CAPIK3CB
Hydrochloric Acid SCHEMBL2920921 0.73 KCNH2 (0.35) KCNH2PIK3CGPIK3CDPIK3CAPIK3CB
SCHEMBL2919816 0.73 PDE10A (0.49) PIK3CGPIK3CDPIK3CAPIK3CBPDE10A
SCHEMBL591477 0.71 ITGB3 (0.45) PPARGPPARA
SCHEMBL2925641 0.71 GRM2 (0.44) AAK1
SCHEMBL2925960 0.69 AKT1 (0.42) AAK1
SCHEMBL5741460 0.69 SIRT2 (0.39)
SCHEMBL590563 0.68 KCNH2 (0.40) KCNH2PIK3CGPIK3CDPIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1560488-A4 ANTIBACTERIAL AGENTS SMITHKLINE BEECHAM CORP (US) 2006-08-02 EP disclosed
EP-1560488-A2 ANTIBACTERIAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2005-08-10 EP disclosed
WO-2004041210-A2 ANTIBACTERIAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2004-05-21 WO disclosed