SCHEMBL5741806

SCHEMBL5741806

Nc1nc(Nc2ccc3nc(-c4cccc(F)c4)cc(N)c3c2)cc(-c2cccc(OCc3ccccc3)c2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.47
EGFR P00533 3/20 0.42
ERBB2 P04626 1/20 0.42
AGPAT2 O15120 1/20 0.41
PDGFRB P09619 1/20 0.41
KDM4E B2RXH2 7/20 0.40
ALDH1A1 P00352 7/20 0.40
MAPT P10636 7/20 0.40
HPGD P15428 7/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
HTT P42858 2/20 0.40
THRB P10828 1/20 0.40
KMT2A Q03164 3/20 0.40
LMNA P02545 3/20 0.40
MEN1 O00255 2/20 0.40
GAA P10253 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.38
ROCK2 O75116 2/20 0.38
MAOB P27338 1/20 0.38
DYRK1B Q9Y463 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5741054 0.94 BACE1 (0.46) BACE1EGFRERBB2AGPAT2KDM4E
SCHEMBL5743131 0.94 BACE1 (0.50) BACE1AGPAT2KDM4EALDH1A1MAPT
SCHEMBL5740722 0.91 BACE1 (0.49) BACE1AGPAT2KDM4EALDH1A1MAPT
SCHEMBL5742899 0.89 AGPAT2 (0.55) BACE1AGPAT2KDM4EALDH1A1MAPT
SCHEMBL5744147 0.88 MCHR1 (0.47) BACE1AGPAT2KDM4EALDH1A1MAPT
SCHEMBL5742375 0.88 MAPT (0.51) BACE1AGPAT2KDM4EALDH1A1MAPT
SCHEMBL5744066 0.88 DOT1L (0.49) BACE1AGPAT2ALDH1A1MAPT
SCHEMBL5740131 0.87 AGPAT2 (0.54) AGPAT2MAPTHPGDHTTTHRB
SCHEMBL5743044 0.87 AGPAT2 (0.50) AGPAT2MAPTTHRBLMNAABCG2
SCHEMBL5742913 0.87 KMT2A (0.43) EGFRERBB2AGPAT2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339706-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2006-04-19 EP disclosed