SCHEMBL5744147

SCHEMBL5744147

Nc1nc(Nc2ccc3nc(-c4ccc(C(F)(F)F)cc4)cc(N)c3c2)cc(-c2cccc(OCc3ccccc3)c2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 3/20 0.47
BACE1 P56817 1/20 0.44
ACP1 P24666 2/20 0.41
AGPAT2 O15120 2/20 0.41
OPRL1 P41146 1/20 0.41
KDM4E B2RXH2 5/20 0.40
ALDH1A1 P00352 5/20 0.40
HPGD P15428 5/20 0.40
MAPT P10636 4/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
HTT P42858 2/20 0.40
THRB P10828 1/20 0.40
GAA P10253 2/20 0.40
LMNA P02545 2/20 0.39
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
SYK P43405 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
GHSR Q92847 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5743033 0.93 MCHR1 (0.47) MCHR1ACP1AGPAT2OPRL1KDM4E
SCHEMBL5743131 0.93 BACE1 (0.50) BACE1AGPAT2KDM4EALDH1A1HPGD
SCHEMBL5741054 0.91 BACE1 (0.46) BACE1ACP1AGPAT2KDM4EALDH1A1
SCHEMBL5742899 0.89 AGPAT2 (0.55) BACE1AGPAT2OPRL1KDM4EALDH1A1
SCHEMBL5742375 0.89 MAPT (0.51) BACE1ACP1AGPAT2KDM4EALDH1A1
SCHEMBL5741806 0.88 BACE1 (0.47) BACE1AGPAT2KDM4EALDH1A1HPGD
SCHEMBL5741066 0.88 ACP1 (0.51) MCHR1ACP1AGPAT2KDM4EALDH1A1
SCHEMBL5742707 0.87 AGPAT2 (0.49) BACE1AGPAT2KDM4EALDH1A1HPGD
SCHEMBL5740722 0.86 BACE1 (0.49) BACE1AGPAT2KDM4EALDH1A1HPGD
SCHEMBL5742700 0.85 MCHR1 (0.52) MCHR1ACP1AGPAT2MAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339706-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2006-04-19 EP disclosed