SCHEMBL5742005

SCHEMBL5742005

Nc1nc(Nc2ccc3nc(-c4ccccc4F)cc(N)c3c2)cc(-c2ccc(Cl)cc2)n1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AGPAT2 O15120 15/20 0.59
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
ROCK2 O75116 2/20 0.42
AURKA O14965 1/20 0.41
PDPK1 O15530 1/20 0.41
TGFBR1 P36897 1/20 0.41
ROCK1 Q13464 1/20 0.41
AURKB Q96GD4 1/20 0.41
ACP1 P24666 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5742912 1.00 AGPAT2 (0.59) AGPAT2TP53MAPTROCK2AURKA
SCHEMBL5743241 0.93 AGPAT2 (0.53) AGPAT2TP53MAPTROCK2AURKA
SCHEMBL5744514 0.92 AGPAT2 (0.47) AGPAT2TP53MAPTROCK2AURKA
SCHEMBL5741931 0.91 AGPAT2 (0.52) AGPAT2ROCK2AURKAPDPK1TGFBR1
SCHEMBL5742556 0.90 AGPAT2 (0.61) AGPAT2TP53MAPTAURKAPDPK1
SCHEMBL5741794 0.89 MCHR1 (0.50) AGPAT2TP53MAPTROCK2AURKA
SCHEMBL5741808 0.89 MCHR1 (0.50) AGPAT2TP53MAPTROCK2AURKA
SCHEMBL5740139 0.88 AGPAT2 (0.60) AGPAT2TP53MAPTROCK2
SCHEMBL5741921 0.86 AGPAT2 (0.51) AGPAT2TP53MAPTROCK2AURKA
SCHEMBL5744254 0.86 AGPAT2 (0.46) AGPAT2ROCK2AURKAPDPK1TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339706-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2006-04-19 EP disclosed