SCHEMBL5744514

SCHEMBL5744514

Nc1nc(Nc2ccc3nc(-c4ccc(F)cc4)cc(N)c3c2)cc(-c2ccccc2F)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGPAT2 O15120 3/20 0.47
ROCK2 O75116 5/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
THRB P10828 1/20 0.43
AURKA O14965 1/20 0.42
PDPK1 O15530 1/20 0.42
TGFBR1 P36897 1/20 0.42
ROCK1 Q13464 1/20 0.42
AURKB Q96GD4 1/20 0.42
CALCA P06881 1/20 0.41
GPR119 Q8TDV5 1/20 0.41
ACP1 P24666 2/20 0.39
ACHE P22303 1/20 0.39
DOT1L Q8TEK3 2/20 0.39
HRH4 Q9H3N8 1/20 0.39
MCHR1 Q99705 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP19A1 P11511 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5743241 0.95 AGPAT2 (0.53) AGPAT2ROCK2LMNATP53MAPT
SCHEMBL5742005 0.92 AGPAT2 (0.59) AGPAT2ROCK2TP53MAPTAURKA
SCHEMBL5742912 0.92 AGPAT2 (0.59) AGPAT2ROCK2TP53MAPTAURKA
SCHEMBL5740176 0.92 AGPAT2 (0.56) AGPAT2ROCK2LMNATP53MAPT
SCHEMBL5741808 0.91 MCHR1 (0.50) AGPAT2ROCK2TP53MAPTAURKA
SCHEMBL5741794 0.91 MCHR1 (0.50) AGPAT2ROCK2TP53MAPTAURKA
SCHEMBL5741921 0.90 AGPAT2 (0.51) AGPAT2ROCK2LMNATP53MAPT
SCHEMBL5744254 0.90 AGPAT2 (0.46) AGPAT2ROCK2AURKAPDPK1TGFBR1
SCHEMBL5742032 0.90 AGPAT2 (0.46) AGPAT2ROCK2AURKAPDPK1TGFBR1
SCHEMBL5740482 0.89 ALOX15 (0.48) AGPAT2ROCK2LMNATP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339706-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2006-04-19 EP disclosed