SCHEMBL5742136

SCHEMBL5742136

C=C[C@H]1CC(=O)C=CN1C(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 2/20 0.41
NFKB2 Q00653 2/20 0.41
RELA Q04206 2/20 0.41
F13A1 P00488 2/20 0.34
TGM2 P21980 2/20 0.34
TGM1 P22735 2/20 0.34
ELANE P08246 1/20 0.34
BUB1 O43683 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
THRB P10828 1/20 0.33
SETD7 Q8WTS6 2/20 0.33
MAPK1 P28482 1/20 0.33
GLA P06280 1/20 0.32
HSD11B1 P28845 1/20 0.32
NPC1 O15118 1/20 0.32
GPR119 Q8TDV5 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4166884 1.00 NFKB1 (0.41) NFKB1NFKB2RELAF13A1TGM2
SCHEMBL13609090 0.82 NFKB1 (0.36) NFKB1NFKB2RELAF13A1TGM2
SCHEMBL758730 0.79 NFKB1 (0.42) NFKB1NFKB2RELAKDM4EMAPT
SCHEMBL760600 0.75 GLA (0.40) NFKB1NFKB2RELAKDM4EMAPT
SCHEMBL3943561 0.75 NR1H2 (0.40) NFKB1NFKB2RELAKDM4EMAPT
SCHEMBL7127132 0.74 PTPN1 (0.41) NFKB1NFKB2RELAKDM4EMAPT
SCHEMBL30534268 0.74 NFKB1 (0.38) NFKB1NFKB2RELAELANEKDM4E
SCHEMBL4152795 0.74 ELANE (0.46) ELANEMAPTNPC1
SCHEMBL4174627 0.72 P2RX7 (0.51) GPR119
SCHEMBL16409264 0.70 P2RX7 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1622871-A1 CYCLIC AMINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 2006-02-08 EP disclosed
WO-2004099143-A1 CYCLIC AMINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 2004-11-18 WO disclosed