SCHEMBL5742340

SCHEMBL5742340

CO/N=C1\C[C@@H](C(=O)NCCc2ccccc2O)N(C(=O)c2ccc(-c3ccccc3)cc2)C1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OXTR P30559 5/20 0.67
AVPR1A P37288 3/20 0.57
HTR1A P08908 1/20 0.40
HTR1B P28222 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
LMNA P02545 2/20 0.37
HIF1A Q16665 1/20 0.37
MMP1 P03956 1/20 0.36
MMP3 P08254 1/20 0.36
MMP7 P09237 1/20 0.36
ALDH1A1 P00352 2/20 0.36
USP2 O75604 1/20 0.36
PKM P14618 1/20 0.36
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
PABPC1 P11940 1/20 0.34
KMT2A Q03164 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4939162 0.87 OXTR (0.73) OXTRAVPR1AHTR1AHTR1BHTR2A
SCHEMBL4944329 0.87 OXTR (0.73) OXTRAVPR1AHTR1AHTR1BHTR2A
SCHEMBL4943696 0.86 OXTR (0.72) OXTRAVPR1ALMNAMMP1MMP3
SCHEMBL4942110 0.85 OXTR (0.71) OXTRAVPR1ALMNAMMP1MMP3
SCHEMBL7164251 0.84 OXTR (0.70) OXTRAVPR1AHTR1AHTR1BHTR2A
SCHEMBL4939792 0.84 OXTR (0.70) OXTRAVPR1AHTR1AHTR1BHTR2A
SCHEMBL7086637 0.84 OXTR (0.70) OXTRAVPR1ALMNAMMP1MMP3
SCHEMBL4943384 0.84 OXTR (0.70) OXTRAVPR1AHTR1AHTR1BHTR2A
SCHEMBL7088615 0.84 OXTR (0.70) OXTRAVPR1AHTR1AHTR1BHTR2A
SCHEMBL4942292 0.84 OXTR (0.70) OXTRAVPR1ALMNAMMP1MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268419-B1 PYRROLIDINE DERIVATIVES USEFUL AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS (AN) 2006-06-21 EP disclosed