SCHEMBL5742875

SCHEMBL5742875

Nc1nc(Nc2ccc3nc(-c4ccc(Cl)cc4)cc(N)c3c2)cc(-c2ccc(C(F)(F)F)cc2)n1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AGPAT2 O15120 10/20 0.57
MCHR1 Q99705 3/20 0.49
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HSD17B10 Q99714 1/20 0.46
ALOX5 P09917 1/20 0.43
ROCK2 O75116 1/20 0.41
NPC1 O15118 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
RAB9A P51151 1/20 0.41
ACP1 P24666 1/20 0.41
TRPV1 Q8NER1 1/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5741991 1.00 AGPAT2 (0.57) AGPAT2MCHR1KDM4EALDH1A1HSD17B10
SCHEMBL5740529 0.95 MCHR1 (0.53) AGPAT2MCHR1ROCK2ACP1TRPV1
SCHEMBL5741862 0.91 AGPAT2 (0.57) AGPAT2MCHR1KDM4EALDH1A1HSD17B10
SCHEMBL5741884 0.91 AGPAT2 (0.52) AGPAT2MCHR1ROCK2ACP1TRPV1
SCHEMBL5741026 0.91 AGPAT2 (0.52) AGPAT2MCHR1ROCK2ACP1TRPV1
SCHEMBL5740460 0.91 MCHR1 (0.50) AGPAT2MCHR1KDM4EROCK2CYP3A4
SCHEMBL5744288 0.89 KDM4E (0.56) AGPAT2MCHR1KDM4EALDH1A1HSD17B10
SCHEMBL5740563 0.89 AGPAT2 (0.52) AGPAT2MCHR1ROCK2ACP1TRPV1
SCHEMBL5740139 0.89 AGPAT2 (0.60) AGPAT2KDM4EALDH1A1HSD17B10ROCK2
SCHEMBL5742700 0.88 MCHR1 (0.52) AGPAT2MCHR1ROCK2ACP1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339706-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2006-04-19 EP disclosed