SCHEMBL5743914

SCHEMBL5743914

CC(C)n1c(C(=O)NCc2ccccc2)nc(Br)c1C=O

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
HPGD P15428 3/20 0.44
HMGCR P04035 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.42
TP53 P04637 1/20 0.41
RORC P51449 1/20 0.41
APOBEC3A P31941 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
ANPEP P15144 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5756156 0.81 HMGCR (0.61) ALDH1A1HPGDHMGCRSMN1; SMN2TP53
SCHEMBL5745018 0.80 HMGCR (0.52) ALDH1A1HMGCRSMN1; SMN2
SCHEMBL5742188 0.80 HMGCR (0.51) ALDH1A1HMGCRSMN1; SMN2
SCHEMBL5742192 0.80 HMGCR (0.51) ALDH1A1HMGCRSMN1; SMN2
SCHEMBL5759558 0.79 HMGCR (0.45) ALDH1A1HMGCRSMN1; SMN2
SCHEMBL5742189 0.78 CYP2C9 (0.49) ALDH1A1HMGCRSMN1; SMN2
SCHEMBL5740858 0.78 HMGCR (0.44) ALDH1A1HMGCRSMN1; SMN2
SCHEMBL5761542 0.74 HMGCR (0.54) ALDH1A1HPGDHMGCRSMN1; SMN2
SCHEMBL5741333 0.74 HMGCR (0.35) ALDH1A1HPGDHMGCRSMN1; SMN2TP53
SCHEMBL20833871 0.69 HPGD (0.55) ALDH1A1HPGDSMN1; SMN2APOBEC3AHDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1727541-A1 IMIDAZOLE-BASED HMG-COA REDUCTASE INHIBITORS Warner-Lambert Company LLC (US) 2006-12-06 EP disclosed
WO-2005079790-A1 IMIDAZOLE-BASED HMG-COA REDUCTASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2005-09-01 WO disclosed