SCHEMBL5745443

SCHEMBL5745443

CCCCCc1ccc(C(=O)N2CC(=CC#N)C[C@H]2C(=O)NC(=O)c2ccc(OC)c(OC)c2)c(=O)o1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CFTR P13569 3/20 0.39
HDAC3 O15379 1/20 0.34
HDAC2 Q92769 1/20 0.34
CNR2 P34972 4/20 0.34
SMPD1 P17405 5/20 0.34
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
ALOX12 P18054 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
POLB P06746 1/20 0.32
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5745439 1.00 CFTR (0.39) CFTRHDAC3HDAC2CNR2SMPD1
SCHEMBL4943701 0.87 EPHX2 (0.39) CFTRCYP2C9POLB
SCHEMBL4943697 0.87 EPHX2 (0.39) CFTRCYP2C9POLB
SCHEMBL4941694 0.78 ALDH1A1 (0.37) CYP2C9L3MBTL1POLBKDM4E
SCHEMBL4941699 0.78 ALDH1A1 (0.37) CYP2C9L3MBTL1POLBKDM4E
SCHEMBL4942929 0.78 EPHX2 (0.40) CFTRCYP2C9POLBMAPK1
SCHEMBL4942950 0.71 EPHX2 (0.39) CFTRCYP2C9L3MBTL1POLB
SCHEMBL4942949 0.71 EPHX2 (0.39) CFTRCYP2C9L3MBTL1POLB
SCHEMBL4945246 0.70 EPHX2 (0.38) CFTRCYP2C9L3MBTL1POLB
SCHEMBL4938441 0.66 MMP1 (0.35) CFTRCNR2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268419-B1 PYRROLIDINE DERIVATIVES USEFUL AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS (AN) 2006-06-21 EP disclosed