SCHEMBL574575

SCHEMBL574575

CC(C)(C)[Si](C)(C)OC[C@H](O)COCCc1ccc(F)cc1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.35
ADRB1 P08588 2/20 0.35
ADRB3 P13945 2/20 0.35
HTT P42858 1/20 0.35
HSP90AB1 P08238 2/20 0.35
ELOVL1 Q9BW60 1/20 0.33
CASR P41180 3/20 0.33
KMT2A Q03164 1/20 0.33
HSP90AA1 P07900 1/20 0.32
NPC1 O15118 1/20 0.32
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL574831 1.00 ADRB2 (0.35) ADRB2ADRB1ADRB3HTTHSP90AB1
SCHEMBL503098 0.84 TAAR1 (0.33) ELOVL1
SCHEMBL503485 0.84 TAAR1 (0.33) ELOVL1
SCHEMBL1245973 0.80 ELOVL1 (0.41) ELOVL1PTGS1PTGS2
SCHEMBL1833345 0.76 ADRB2 (0.36) ADRB2ADRB1ADRB3CASRKMT2A
SCHEMBL1842362 0.76 ADRB2 (0.36) ADRB2ADRB1ADRB3CASRKMT2A
SCHEMBL574862 0.75 CYP1A2 (0.40) ADRB2ADRB1ADRB3HSP90AA1
SCHEMBL502775 0.75 ADRB2 (0.36) ADRB2ADRB1ADRB3HTTCASR
SCHEMBL502893 0.75 ADRB2 (0.36) ADRB2ADRB1ADRB3HTTCASR
SCHEMBL502774 0.75 ADRB2 (0.36) ADRB2ADRB1ADRB3HTTCASR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2600853-A1 COMBINATIONS COMPRISING ATYPICAL ANTIPSYCHOTICS AND TAAR1 AGONISTS F.HOFFMANN-LA ROCHE AG (CH) 2013-06-12 EP disclosed
WO-2012016879-A1 COMBINATIONS COMPRISING ATYPICAL ANTIPSYCHOTICS AND TAAR1 AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2012-02-09 WO disclosed