SCHEMBL5745992

SCHEMBL5745992

O=C(CBr)c1ccc(OCCF)cc1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 8/20 0.58
PTPN1 P18031 5/20 0.53
MAPT P10636 1/20 0.53
L3MBTL1 Q9Y468 2/20 0.51
ALDH1A1 P00352 1/20 0.50
NPC1 O15118 1/20 0.46
THRA P10827 1/20 0.46
THRB P10828 1/20 0.46
MMP1 P03956 1/20 0.45
GAA P10253 2/20 0.45
PKM P14618 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9786122 0.87 GSK3B (0.59) GSK3BPTPN1MAPTL3MBTL1ALDH1A1
SCHEMBL15018952 0.86 GSK3B (0.58) GSK3BPTPN1MAPTL3MBTL1NPC1
SCHEMBL1373155 0.82 GSK3B (0.58) GSK3BPTPN1MAPTL3MBTL1NPC1
SCHEMBL5055145 0.82 L3MBTL1 (0.65) GSK3BMAPTL3MBTL1ALDH1A1NPC1
SCHEMBL11728169 0.82 GSK3B (0.58) GSK3BPTPN1MAPTL3MBTL1GAA
SCHEMBL5057170 0.82 L3MBTL1 (0.70) GSK3BPTPN1MAPTL3MBTL1ALDH1A1
SCHEMBL2985635 0.81 GSK3B (0.53) GSK3BPTPN1MAPTL3MBTL1GAA
Bromide SCHEMBL931587 0.81 GSK3B (0.56) GSK3BPTPN1MAPTL3MBTL1NPC1
SCHEMBL2953290 0.81 GSK3B (0.66) GSK3BPTPN1MAPTL3MBTL1THRA
SCHEMBL22007778 0.80 GSK3B (0.51) GSK3BPTPN1MAPTL3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0842923-B1 PYRROLE DERIVATIVES AND MEDICINAL COMPOSITION NIPPON SHINYAKU CO LTD (JP) 2006-03-01 EP disclosed
US-6172102-B1 POLLAKIURIA OR URINARY INCONTINENCE NIPPON SHINYAKU CO., LTD. (JP) 2001-01-09 US disclosed
US-5998459-A INCOTINENCE THERAPY NIPPON SHINYAKU CO., LTD. (JP) 1999-12-07 US disclosed
EP-0842923-A1 PYRROLE DERIVATIVES AND MEDICINAL COMPOSITION NIPPON SHINYAKU COMPANY, LIMITED (JP) 1998-05-20 EP disclosed