SCHEMBL5746334

SCHEMBL5746334

NCCCOc1cccc2oc(=O)c3ccccc3c12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 2/20 0.53
KCNA3 P22001 2/20 0.43
ALDH1A1 P00352 3/20 0.40
GLA P06280 1/20 0.40
CDC25A P30304 1/20 0.40
CDC25B P30305 1/20 0.40
CDC25C P30307 1/20 0.40
LOXL2 Q9Y4K0 1/20 0.40
CYP2A6 P11509 1/20 0.40
MAOA P21397 1/20 0.39
BCHE P06276 2/20 0.39
ACHE P22303 2/20 0.39
KDM4E B2RXH2 3/20 0.39
APEX1 P27695 1/20 0.38
BCL2 P10415 1/20 0.38
BCL2L1 Q07817 1/20 0.38
MCL1 Q07820 1/20 0.38
BAD Q92934 1/20 0.38
GAA P10253 1/20 0.38
KMT2A Q03164 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5749087 0.93 HTR1B (0.51) HTR1BKCNA3ALDH1A1GLACDC25A
SCHEMBL5747324 0.85 HTR1B (0.58) HTR1BKCNA3CDC25ACDC25BCDC25C
SCHEMBL5746372 0.83 MAOA (0.60) HTR1BKCNA3ALDH1A1GLACYP2A6
SCHEMBL5746754 0.82 HRH1 (0.56) HTR1BKCNA3CDC25ACDC25BCDC25C
SCHEMBL10652572 0.81 CYP2A6 (0.55) ALDH1A1CYP2A6MAOABCHEACHE
SCHEMBL5748119 0.81 HTR1B (0.55) HTR1BALDH1A1CYP2A6MAOAKDM4E
SCHEMBL5749229 0.80 HTR1B (0.58) HTR1BCDC25ACDC25BCDC25CCYP2A6
SCHEMBL5748123 0.79 HTR1B (0.59) HTR1BCDC25ACDC25BCDC25CCYP2A6
SCHEMBL10593907 0.75 MAOA (0.66) ALDH1A1CYP2A6MAOABCHEACHE
SCHEMBL31241235 0.74 BCHE (0.37) ALDH1A1GLAMAOABCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP claimed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO claimed
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP disclosed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO disclosed