SCHEMBL5746754

SCHEMBL5746754

CNCCCOc1cccc2oc(=O)c3ccccc3c12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 3/20 0.56
SLC6A4 P31645 2/20 0.56
HTR1B P28222 5/20 0.50
HTR1D P28221 1/20 0.50
ADRB2 P07550 1/20 0.42
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
CDC25A P30304 1/20 0.41
CDC25B P30305 1/20 0.41
CDC25C P30307 1/20 0.41
KCNA3 P22001 1/20 0.40
HTR6 P50406 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5748119 0.96 HTR1B (0.55) HRH1SLC6A4HTR1BHTR1DKDM4E
SCHEMBL5749229 0.87 HTR1B (0.58) HTR1BHTR1DADRB2KDM4ELMNA
SCHEMBL5745016 0.86 SLC6A4 (0.61) HRH1SLC6A4HTR1BHTR1DADRB2
SCHEMBL5748123 0.86 HTR1B (0.59) HTR1BHTR1DADRB2KDM4ELMNA
SCHEMBL5748462 0.84 MAOA (0.59) HRH1SLC6A4HTR1BHTR1DCYP3A4
SCHEMBL5746334 0.82 HTR1B (0.53) HTR1BCYP1A2CYP2C9L3MBTL1KDM4E
SCHEMBL5744798 0.82 HTR1B (0.60) HRH1SLC6A4HTR1BHTR1DADRB2
SCHEMBL5749087 0.81 HTR1B (0.51) HTR1BTP53CYP1A2CYP2C9L3MBTL1
SCHEMBL10652572 0.80 CYP2A6 (0.55) TSHRL3MBTL1KDM4EMAPT
SCHEMBL5749472 0.80 MAOA (0.61) HRH1SLC6A4HTR1BHTR1DCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP claimed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO claimed