SCHEMBL5746469

SCHEMBL5746469

COCCOc1cccc(C(=O)CBr)c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.53
KMT2A Q03164 2/20 0.51
SMPD1 P17405 3/20 0.48
THRA P10827 1/20 0.47
THRB P10828 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.46
LMNA P02545 1/20 0.46
MAPK1 P28482 1/20 0.46
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 1/20 0.45
PTPN1 P18031 2/20 0.45
MEN1 O00255 1/20 0.44
TAAR1 Q96RJ0 1/20 0.44
NR1H4 Q96RI1 1/20 0.44
NPC1 O15118 1/20 0.44
POLB P06746 1/20 0.44
RAB9A P51151 1/20 0.44
BLM P54132 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5057129 0.86 KMT2A (0.69) GSK3BKMT2ASMPD1THRATHRB
SCHEMBL24611877 0.86 KMT2A (0.56) KMT2ASMPD1THRATHRBL3MBTL1
SCHEMBL5051428 0.85 THRB (0.60) GSK3BKMT2ASMPD1THRATHRB
SCHEMBL28294885 0.84 L3MBTL1 (0.57) KMT2ASMPD1L3MBTL1LMNAMAPK1
SCHEMBL8085066 0.84 THRB (0.66) GSK3BKMT2ASMPD1THRATHRB
SCHEMBL5746204 0.83 GSK3B (0.54) GSK3BKMT2ASMPD1THRATHRB
SCHEMBL5260954 0.83 GSK3B (0.54) GSK3BKMT2ASMPD1THRATHRB
SCHEMBL920107 0.83 HPGD (0.54) GSK3BKMT2AL3MBTL1LMNAMAPK1
SCHEMBL1665041 0.83 KMT2A (0.73) KMT2ASMPD1NR1H4
SCHEMBL1665037 0.83 KMT2A (0.55) KMT2ASMPD1THRBL3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0842923-B1 PYRROLE DERIVATIVES AND MEDICINAL COMPOSITION NIPPON SHINYAKU CO LTD (JP) 2006-03-01 EP disclosed
CN-1349796-A Pyrrole derivatives and medicine composition NIPPON SHINYAKU CO LTD (JP) 2002-05-22 CN disclosed
US-6172102-B1 POLLAKIURIA OR URINARY INCONTINENCE NIPPON SHINYAKU CO., LTD. (JP) 2001-01-09 US disclosed
US-5998459-A INCOTINENCE THERAPY NIPPON SHINYAKU CO., LTD. (JP) 1999-12-07 US disclosed
EP-0842923-A1 PYRROLE DERIVATIVES AND MEDICINAL COMPOSITION NIPPON SHINYAKU COMPANY, LIMITED (JP) 1998-05-20 EP disclosed