SCHEMBL5746783

SCHEMBL5746783

CNc1nc(C)cc(N2CCCc3ccccc32)n1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.62
ROCK1 Q13464 2/20 0.49
TUBB4A P04350 2/20 0.45
TUBB P07437 2/20 0.45
TUBA3C P0DPH7 2/20 0.45
TUBA1B P68363 2/20 0.45
TUBA4A P68366 2/20 0.45
TUBB4B P68371 2/20 0.45
TUBB3 Q13509 2/20 0.45
TUBB2A Q13885 2/20 0.45
TUBB8 Q3ZCM7 2/20 0.45
TUBA3E Q6PEY2 2/20 0.45
TUBA1A Q71U36 2/20 0.45
TUBA1C Q9BQE3 2/20 0.45
TUBB6 Q9BUF5 2/20 0.45
TUBB2B Q9BVA1 2/20 0.45
TUBB1 Q9H4B7 2/20 0.45
SMN1; SMN2 Q16637 4/20 0.44
ALDH1A1 P00352 4/20 0.44
MEN1 O00255 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9377990 0.92 NUDT1 (0.52) NUDT1ROCK1SMN1; SMN2ALDH1A1MEN1
Hydrochloric Acid SCHEMBL5749583 0.82 NUDT1 (0.69) NUDT1ROCK1TUBB4ATUBBTUBA3C
SCHEMBL5750076 0.81 ROCK1 (0.67) NUDT1ROCK1TUBB4ATUBBTUBA3C
SCHEMBL5747568 0.79 NUDT1 (0.65) NUDT1ROCK1SMN1; SMN2ALDH1A1MEN1
SCHEMBL9004353 0.78 NUDT1 (0.51) NUDT1ROCK1TUBB4ATUBBTUBA3C
SCHEMBL9382651 0.78 NUDT1 (0.46) NUDT1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL24265310 0.75 ROCK1 (0.59) NUDT1ROCK1SMN1; SMN2ALDH1A1MEN1
SCHEMBL7077159 0.74 ROCK1 (0.61) NUDT1ROCK1SMN1; SMN2ALDH1A1MEN1
SCHEMBL17033290 0.71 ROCK1 (0.62) NUDT1ROCK1TUBB4ATUBBTUBA3C
Hydrochloric Acid SCHEMBL5746691 0.70 NUDT1 (0.68) NUDT1ROCK1SMN1; SMN2ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901474-B1 ARYL PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2006-04-19 EP disclosed
EP-1321169-A1 Combination of a serotonin receptor antagonist with a histidine decarboxylase inhibitor as a medicament Biofrontera Pharmaceuticals AG (DE) 2003-06-25 EP disclosed
CN-1109675-C Aryl pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2003-05-28 CN disclosed
US-5958934-A 5-HT 2B ANTAGONIST SYNTEX (U.S.A.) INC. (US) 1999-09-28 US disclosed
US-5952331-A SELECTIVE 5HT2B ANTAGONISTS; SEROTONIN RECEPTOR ANTAGONIST; TREATING DISORDERS OF THE GASTROINTESTINAL TRACK, RESTENOSIS, ASTHMA AND OBSTRUCTIVE AIRWAY DISEASE, PROSTATIC HYPERPLASIA, GENERALIZED ANXIETY, PANIC DISORDER SYNTEX (USA) INC. (US) 1999-09-14 US disclosed
CN-1223641-A Aryl pyrimidine derivatives HOFFMANN LA ROCHE (CH) 1999-07-21 CN disclosed
US-5863924-A Aryl pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1999-01-26 US disclosed