SCHEMBL9004353

SCHEMBL9004353

CNc1nc(C)nc(N2CCCc3ccccc32)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.51
MAPT P10636 7/20 0.48
ALDH1A1 P00352 6/20 0.48
LMNA P02545 4/20 0.48
SMN1; SMN2 Q16637 4/20 0.48
MAPK1 P28482 3/20 0.48
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
TP53 P04637 2/20 0.48
ALOX15 P16050 1/20 0.48
JAK2 O60674 1/20 0.46
JAK3 P52333 1/20 0.46
PTK2 Q05397 1/20 0.46
ROCK1 Q13464 1/20 0.44
HTT P42858 1/20 0.44
TUBB4A P04350 1/20 0.43
TUBB P07437 1/20 0.43
TUBA3C P0DPH7 1/20 0.43
TUBA1B P68363 1/20 0.43
TUBA4A P68366 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9004433 0.80 NPC1 (0.52) NUDT1MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL5746783 0.78 NUDT1 (0.62) NUDT1MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL9004357 0.76 NPC1 (0.60) NUDT1MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL2900973 0.74 EPHX2 (0.47) ALDH1A1JAK2JAK3PTK2ROCK1
SCHEMBL13238876 0.74 EPHX2 (0.66) MAPTEPHX2
SCHEMBL5750076 0.74 ROCK1 (0.67) NUDT1MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL27424682 0.74 NUDT1 (0.57) NUDT1MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL17486069 0.73 JAK2 (0.53) NUDT1MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL5063173 0.73 JAK2 (0.53) NUDT1MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL9377990 0.72 NUDT1 (0.52) NUDT1MAPTALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5574037-A MODULATED BY SINO-ATRIAL NODE, ANTIISCHEMIC AGENT IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1996-11-12 US disclosed
EP-0431856-B1 Heterocyclic compounds ZENECA LTD (GB) 1995-07-12 EP disclosed
US-5332737-A Cardiovascular disorders IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-07-26 US disclosed
EP-0431856-A2 Heterocyclic compounds ZENECA LIMITED (GB) 1991-06-12 EP disclosed