SCHEMBL5749013

SCHEMBL5749013

NC(=O)c1cccc2cc[c]nc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 17/20 0.58
PARP2 Q9UGN5 2/20 0.44
PARP3 Q9Y6F1 2/20 0.44
PLK4 O00444 1/20 0.42
CHEK1 O14757 1/20 0.42
AURKA O14965 1/20 0.42
DAPK3 O43293 1/20 0.42
MAP4K4 O95819 1/20 0.42
CSF1R P07333 1/20 0.42
RET P07949 1/20 0.42
FGFR1 P11362 1/20 0.42
PDGFRA P16234 1/20 0.42
LTK P29376 1/20 0.42
KDR P35968 1/20 0.42
MAP2K2 P36507 1/20 0.42
FLT3 P36888 1/20 0.42
CSNK1A1 P48729 1/20 0.42
PRKX P51817 1/20 0.42
CDK5 Q00535 1/20 0.42
MAP2K1 Q02750 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8487622 0.84 ALDH1A1 (0.47) PARP1KDM4EALDH1A1
SCHEMBL16289662 0.79 KDM4E (0.46) PARP1KDM4EALDH1A1GAA
SCHEMBL29923839 0.74 PARP1 (1.00) PARP1GAA
SCHEMBL422282 0.74 PARP1 (1.00) PARP1GAA
SCHEMBL29959688 0.73 PARP1 (1.00) PARP1PLK4MAP4K4FLT3KDM4E
SCHEMBL460456 0.73 PARP1 (1.00) PARP1PLK4MAP4K4FLT3KDM4E
SCHEMBL29923346 0.73 PARP1 (1.00) PARP1PLK4MAP4K4FLT3KDM4E
SCHEMBL5749771 0.72 KDM4E (0.42) PARP1PLK4CHEK1AURKADAPK3
Hydrochloric Acid SCHEMBL18094592 0.71 PARP1 (0.96) PARP1PLK4MAP4K4FLT3KDM4E
Hydrochloric Acid SCHEMBL29933479 0.71 PARP1 (0.96) PARP1PLK4MAP4K4FLT3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060293503-A1 Polyaminopyridines and method for producing same SUMITOMO SEIKA CHEMICALS CO., LTD (JP) 2006-12-28 US disclosed
EP-1669390-A1 POLYAMINOPYRIDINES AND METHOD FOR PRODUCING SAME SUMITOMO SEIKA CHEMICALS CO., LTD. (JP) 2006-06-14 EP disclosed