SCHEMBL5749679

SCHEMBL5749679

CN(C)CCNCCCc1nc2c(c(=O)n1Cc1ccccc1)CCC2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
PABPC1 P11940 1/20 0.43
EIF4H Q15056 1/20 0.43
PDE4A P27815 3/20 0.42
PDE4B Q07343 3/20 0.42
PDE4C Q08493 3/20 0.42
PDE4D Q08499 3/20 0.42
RAD52 P43351 1/20 0.41
GAA P10253 2/20 0.41
MAPT P10636 2/20 0.41
MAPK1 P28482 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HRH3 Q9Y5N1 3/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
MITF O75030 1/20 0.40
POLB P06746 1/20 0.39
HTT P42858 1/20 0.39
HRH2 P25021 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5749676 0.80 HPGD (0.47) MEN1KMT2APDE4APDE4BPDE4C
SCHEMBL4029525 0.80 PDE4A (0.51) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL5750358 0.77 KIF11 (0.42) MEN1KMT2APDE4APDE4BPDE4C
SCHEMBL5144677 0.77 PDE4A (0.49) MEN1KMT2APDE4APDE4BPDE4C
SCHEMBL5555021 0.77 PDE4A (0.49) MEN1KMT2APDE4APDE4BPDE4C
SCHEMBL5738140 0.77 PDE4B (0.69) KMT2APDE4APDE4BPDE4CPDE4D
SCHEMBL5784852 0.77 PDE4A (0.49) MEN1KMT2APDE4APDE4BPDE4C
SCHEMBL4028286 0.77 MEN1 (0.46) MEN1KMT2APABPC1EIF4HRAD52
SCHEMBL5740040 0.76 MEN1 (0.41) MEN1KMT2APDE4APDE4BPDE4C
SCHEMBL5144517 0.74 KIF11 (0.45) MEN1KMT2APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551812-A4 MITOTIC KINESIN INHIBITORS MERCK & CO INC (US) 2006-01-04 EP disclosed
EP-1551812-A2 MITOTIC KINESIN INHIBITORS Merck & Co., Inc. (US) 2005-07-13 EP disclosed
WO-2003049678-A2 MITOTIC KINESIN INHIBITORS MERCK & CO., INC. (US) 2003-06-19 WO disclosed