SCHEMBL5749784

SCHEMBL5749784

CC(F)(F)c1ccc(CC(N)C(O)c2ccc(F)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.41
AOC3 Q16853 1/20 0.36
GRB2 P62993 1/20 0.35
PDE2A O00408 1/20 0.34
MMP2 P08253 1/20 0.33
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
PTPN1 P18031 1/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
KIF11 P52732 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5751727 0.88 TRPA1 (0.39) TRPA1GRB2NOS3NOS1NOS2
SCHEMBL6578585 0.88 TRPA1 (0.39) TRPA1GRB2NOS3NOS1NOS2
SCHEMBL5750053 0.88 TRPA1 (0.39) TRPA1GRB2NOS3NOS1NOS2
Hydrochloric Acid SCHEMBL5751082 0.87 TACR1 (0.39) TRPA1NOS3NOS1NOS2
SCHEMBL5749249 0.86 TRPA1 (0.47) TRPA1AOC3MMP2
SCHEMBL5750636 0.84 HTR2A (0.47) LMNA
SCHEMBL5752240 0.82 TRPA1 (0.49) TRPA1AOC3ESR1ESR2
SCHEMBL5753279 0.80 TRPA1 (0.42) TRPA1AOC3MMP2
SCHEMBL5749920 0.80 KMT2A (0.43) GRB2ESR1PTPN1LMNA
SCHEMBL5751556 0.79 CASR (0.44) TRPA1PTPN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6982348-B2 Aminoethanol derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2006-01-03 US disclosed
US-20040127574-A1 Aminoethanol derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-07-01 US disclosed
EP-1362846-A1 AMINOETHANOL DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 2003-11-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040127574-A1 Aminoethanol derivatives CETP, LCAT, MTTP TRPA1 3461/4885AOC3 2703/4885GRB2 1627/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.