SCHEMBL5749249

SCHEMBL5749249

NC(Cc1ccc(F)cc1)C(O)c1ccc(F)cc1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.47
AOC3 Q16853 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.40
MMP2 P08253 2/20 0.40
TAAR1 Q96RJ0 1/20 0.38
HTT P42858 1/20 0.37
IDO1 P14902 3/20 0.36
AGXT P21549 1/20 0.36
TDO2 P48775 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5753279 0.93 TRPA1 (0.42) TRPA1AOC3LOXL2MMP2TAAR1
SCHEMBL5752240 0.92 TRPA1 (0.49) TRPA1AOC3TAAR1HTTIDO1
SCHEMBL5750053 0.89 TRPA1 (0.39) TRPA1TAAR1IDO1
SCHEMBL6578585 0.89 TRPA1 (0.39) TRPA1TAAR1IDO1
SCHEMBL5751727 0.89 TRPA1 (0.39) TRPA1TAAR1IDO1
SCHEMBL5752285 0.87 CYP1A2 (0.55) AOC3HTT
SCHEMBL5751018 0.87 MAOA (0.44) TRPA1LOXL2
Hydrochloric Acid SCHEMBL5751082 0.87 TACR1 (0.39) TRPA1TAAR1IDO1
SCHEMBL5749784 0.86 TRPA1 (0.41) TRPA1AOC3MMP2
SCHEMBL5751556 0.85 CASR (0.44) TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6982348-B2 Aminoethanol derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2006-01-03 US disclosed
US-20040127574-A1 Aminoethanol derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-07-01 US disclosed
EP-1362846-A1 AMINOETHANOL DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 2003-11-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040127574-A1 Aminoethanol derivatives CETP, LCAT, MTTP TRPA1 3461/4885AOC3 2703/4885LOXL2 2439/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.