SCHEMBL5751225

SCHEMBL5751225

Cc1ccc(C(C#N)(CCCN2CCN(CCOc3ccc(F)cc3)CC2)C(C)C)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 3/20 0.47
ALDH1A1 P00352 2/20 0.47
USP2 O75604 1/20 0.47
HPGD P15428 1/20 0.47
DRD2 P14416 3/20 0.47
DRD3 P35462 3/20 0.47
DRD1 P21728 2/20 0.47
DRD5 P21918 1/20 0.47
SIGMAR1 Q99720 2/20 0.43
HTR1A P08908 2/20 0.43
HTR2A P28223 2/20 0.43
LMNA P02545 3/20 0.43
LTA4H P09960 1/20 0.43
MEN1 O00255 1/20 0.43
HTT P42858 1/20 0.43
KMT2A Q03164 1/20 0.43
HRH3 Q9Y5N1 1/20 0.42
KCNA5 P22460 1/20 0.42
HRH1 P35367 1/20 0.42
TMEM97 Q5BJF2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5752298 0.96 ALDH1A1 (0.51) CACNA1BALDH1A1USP2HPGDDRD2
SCHEMBL5754140 0.92 MEN1 (0.48) CACNA1BALDH1A1USP2HPGDDRD2
SCHEMBL5752620 0.92 CACNA1B (0.51) CACNA1BALDH1A1USP2HPGDDRD2
SCHEMBL5754925 0.91 CACNA1B (0.49) CACNA1BALDH1A1USP2HPGDDRD2
SCHEMBL5753684 0.91 CACNA1B (0.47) CACNA1BALDH1A1USP2HPGDDRD2
SCHEMBL5755060 0.91 DRD2 (0.52) CACNA1BALDH1A1USP2HPGDDRD2
SCHEMBL2866236 0.91 CACNA1B (0.52) CACNA1BALDH1A1USP2HPGDDRD2
Hydrochloric Acid SCHEMBL5754015 0.90 CACNA1B (0.53) CACNA1BALDH1A1USP2HPGDDRD2
SCHEMBL5753216 0.89 CACNA1B (0.46) CACNA1BALDH1A1USP2HPGDDRD2
SCHEMBL5751939 0.89 CACNA1B (0.46) CACNA1BALDH1A1USP2HPGDDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP claimed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US claimed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP claimed
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP disclosed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US disclosed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP disclosed