SCHEMBL5752014

SCHEMBL5752014

CCOC(=O)COc1cc(F)ccc1OCCO

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
KMT2A Q03164 4/20 0.48
GAA P10253 2/20 0.48
KDM4E B2RXH2 2/20 0.48
USP2 O75604 1/20 0.47
MAPT P10636 2/20 0.44
LMNA P02545 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HPGD P15428 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
PTPN1 P18031 1/20 0.43
NPC1 O15118 1/20 0.43
S1PR4 O95977 1/20 0.43
ITGA4 P13612 1/20 0.43
S1PR1 P21453 1/20 0.43
MAPK1 P28482 1/20 0.43
RAB9A P51151 1/20 0.43
TLR9 Q9NR96 1/20 0.43
MEN1 O00255 2/20 0.43
CXCR1 P25024 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30717645 0.86 USP2 (0.61) ALDH1A1KMT2AGAAKDM4EUSP2
SCHEMBL9631971 0.82 KMT2A (0.54) ALDH1A1KMT2AGAAKDM4EMAPT
SCHEMBL13239750 0.81 LMNA (0.58) ALDH1A1KMT2AGAAKDM4EUSP2
SCHEMBL13603359 0.81 FFAR1 (0.50) ALDH1A1GAAUSP2MAPTLMNA
SCHEMBL29536561 0.81 LMNA (0.58) ALDH1A1KMT2AGAAKDM4EUSP2
SCHEMBL2226476 0.81 HTR2C (0.44) ALDH1A1KMT2AGAAKDM4EMAPT
SCHEMBL18688117 0.79 HTR2C (0.46) ALDH1A1KMT2AGAAKDM4EUSP2
SCHEMBL9632944 0.79 HTR2C (0.46) ALDH1A1KMT2AGAAKDM4EUSP2
SCHEMBL15941407 0.79 F9 (0.51) ALDH1A1KMT2AGAAKDM4EUSP2
SCHEMBL5529143 0.79 PKM (0.66) ALDH1A1KMT2AGAAKDM4EUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP disclosed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US disclosed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP disclosed