SCHEMBL5753072

SCHEMBL5753072

CCCCC(C#N)(CCC=O)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EBP Q15125 1/20 0.50
SIGMAR1 Q99720 1/20 0.50
CCR1 P32246 4/20 0.36
DRD2 P14416 2/20 0.36
DRD4 P21917 2/20 0.36
OPRM1 P35372 2/20 0.36
DRD3 P35462 2/20 0.36
CYP2D6 P10635 1/20 0.36
KIF11 P52732 1/20 0.35
CHRM3 P20309 4/20 0.34
LMNA P02545 1/20 0.34
TSHR P16473 2/20 0.33
ATM Q13315 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
PTGS2 P35354 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM1 P11229 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5753670 0.91 EBP (0.43) EBPSIGMAR1CCR1DRD2DRD4
SCHEMBL51900 0.87 EBP (0.59) EBPSIGMAR1CCR1DRD2DRD4
SCHEMBL3888982 0.87 EBP (0.51) EBPSIGMAR1CCR1DRD2DRD4
SCHEMBL5754187 0.86 CCR1 (0.40) EBPSIGMAR1CCR1DRD2DRD4
SCHEMBL5756879 0.79 CYP2D6 (0.37) EBPSIGMAR1DRD2DRD4OPRM1
SCHEMBL7355570 0.79 ALDH1A1 (0.42) EBPSIGMAR1DRD2DRD4OPRM1
SCHEMBL11448920 0.78 EBP (0.51) EBPSIGMAR1CCR1DRD2DRD4
SCHEMBL11479026 0.78 EBP (0.51) EBPSIGMAR1CCR1DRD2DRD4
SCHEMBL11646369 0.78 SIGMAR1 (0.64) EBPSIGMAR1CCR1DRD2DRD4
SCHEMBL7313305 0.78 EBP (0.42) EBPSIGMAR1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP disclosed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US disclosed
CN-1310709-A N, N-substituted cyclic amine derivatives EISAI CO LTD (JP) 2001-08-29 CN disclosed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP disclosed