SCHEMBL5753172

SCHEMBL5753172

CC(C)C(C#N)(CCCN1CCN(CCOc2ccc(F)cc2OCCO)CC1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 3/20 0.47
LMNA P02545 2/20 0.45
POLB P06746 2/20 0.45
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
HTT P42858 1/20 0.40
CACNA1G O43497 1/20 0.40
CCR1 P32246 1/20 0.40
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 3/20 0.37
EBP Q15125 2/20 0.37
SIGMAR1 Q99720 2/20 0.37
CCR3 P51677 1/20 0.37
HTR7 P34969 2/20 0.36
HTR1A P08908 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5753652 0.91 CACNA1B (0.56) CACNA1BLMNAKDM4EALDH1A1
SCHEMBL5754627 0.90 CACNA1B (0.46) CACNA1BLMNAMEN1KMT2AHTT
SCHEMBL5751383 0.89 CACNA1B (0.48) CACNA1BLMNAPOLBMEN1KMT2A
SCHEMBL5753788 0.87 CACNA1G (0.46) CACNA1BMEN1KMT2ACACNA1GCCR1
SCHEMBL5751449 0.85 KDM4E (0.48) CACNA1BLMNAPOLBMEN1KMT2A
SCHEMBL2866236 0.83 CACNA1B (0.52) CACNA1BLMNAMEN1KMT2ACACNA1G
SCHEMBL5753351 0.83 CACNA1B (0.52) CACNA1BLMNAMEN1KMT2AHTT
Hydrochloric Acid SCHEMBL5754015 0.82 CACNA1B (0.53) CACNA1BLMNAMEN1KMT2ACACNA1G
SCHEMBL5753291 0.81 CACNA1B (0.48) CACNA1BLMNAPOLBMEN1KMT2A
SCHEMBL5749773 0.81 CACNA1B (0.48) CACNA1BLMNAPOLBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP claimed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US claimed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP claimed
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP disclosed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US disclosed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP disclosed