SCHEMBL5757189

SCHEMBL5757189

O=S(=O)(c1ccc(F)cc1CCCl)c1ccc(F)cc1CCCl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39
HTR2A P28223 2/20 0.36
HTR2C P28335 2/20 0.36
AKR1B1 P15121 2/20 0.35
MMP1 P03956 1/20 0.35
MMP2 P08253 1/20 0.35
MMP3 P08254 1/20 0.35
MMP9 P14780 1/20 0.35
MMP12 P39900 1/20 0.35
MMP13 P45452 1/20 0.35
MMP14 P50281 1/20 0.35
KDM4E B2RXH2 1/20 0.34
PTGES2 Q9H7Z7 2/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
KMT2A Q03164 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3948236 0.85 PSEN1 (0.41) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5957559 0.79 CNR2 (0.40) AKR1B1PTGES2KMT2ATSHRMAPK1
SCHEMBL8978666 0.79 KDM4E (0.40) KDM4EPTGDR2KMT2ATSHRMAPK1
SCHEMBL4118278 0.79 KDM4E (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL9820115 0.78 TAAR1 (0.36) PTGES2KMT2A
SCHEMBL31356938 0.77 CYP2D6 (0.46) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL31356939 0.77 PSEN1 (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4436410 0.77 CYP2D6 (0.46) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4437847 0.77 PSEN1 (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL31356935 0.75 CYP2D6 (0.46) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP disclosed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US disclosed