SCHEMBL5757703

SCHEMBL5757703

c1ccc(C(Cc2nc(COc3ccc(CCCn4ccnc4)cc3)co2)c2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HMOX1 P09601 2/20 0.53
GLA P06280 1/20 0.45
HTT P42858 1/20 0.45
CYP19A1 P11511 2/20 0.45
LTA4H P09960 1/20 0.43
KMT2A Q03164 1/20 0.43
ATP4A P20648 1/20 0.42
ATP4B P51164 1/20 0.42
CACNA1B Q00975 1/20 0.42
TBXAS1 P24557 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5758029 0.89 HMOX1 (0.59) HMOX1GLAHTTCYP19A1LTA4H
SCHEMBL5762170 0.88 HMOX1 (0.58) HMOX1GLAHTTCYP19A1LTA4H
SCHEMBL5756471 0.83 HMOX1 (0.48) HMOX1CYP19A1TBXAS1
SCHEMBL5760668 0.83 FFAR1 (0.59) HMOX1HTTLTA4HATP4AATP4B
SCHEMBL5760800 0.81 PPARG (0.49) HMOX1HTTLTA4HKMT2AATP4A
SCHEMBL5761313 0.81 HMOX1 (0.48) HMOX1GLAHTTCYP19A1LTA4H
SCHEMBL5761017 0.81 HMOX1 (0.49) HMOX1GLAHTTCYP19A1LTA4H
SCHEMBL5756734 0.81 HMOX1 (0.47) HMOX1CYP19A1ATP4AATP4B
SCHEMBL5760394 0.81 HMOX1 (0.47) HMOX1CYP19A1LTA4HKMT2AATP4A
SCHEMBL5759974 0.80 HMOX1 (0.62) HMOX1HTTCYP19A1LTA4HKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1270571-B1 Heterocyclic compounds, their production and use TAKEDA PHARMACEUTICAL (JP) 2006-09-06 EP disclosed
EP-1270571-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-01-02 EP disclosed
US-6211215-B1 AROMATIC HETEROCYCLIC COMPOUND WITH AZOLE COMPOUND TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US disclosed