SCHEMBL5758099

SCHEMBL5758099

CCn1nc(C2=C(c3cn(CCCN4CCOCC4)c4ccccc34)C(=O)NC2=O)c2cc(Cl)ccc21

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 18/20 0.67
PRKACA P17612 2/20 0.58
PRKACG P22612 2/20 0.58
PRKACB P22694 2/20 0.58
PRKCG P05129 2/20 0.58
PRKCB P05771 2/20 0.58
PRKCA P17252 2/20 0.58
KCNH2 Q12809 1/20 0.58
KDR P35968 2/20 0.52
QPCT Q16769 2/20 0.52
IDH1 O75874 1/20 0.51
CCNB2 O95067 1/20 0.50
CDK1 P06493 1/20 0.50
PDGFRB P09619 1/20 0.50
CCNB1 P14635 1/20 0.50
PDGFRA P16234 1/20 0.50
PRKCE Q02156 1/20 0.50
PRKCD Q05655 1/20 0.50
CAMK2B Q13554 1/20 0.50
CAMK2G Q13555 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5756212 0.93 GSK3B (0.56) GSK3BPRKCGPRKCBPRKCAKCNH2
SCHEMBL5758425 0.92 GSK3B (0.58) GSK3BPRKACAPRKACGPRKACBPRKCG
SCHEMBL5758352 0.87 GSK3B (0.58) GSK3BPRKACAPRKACGPRKACBPRKCG
SCHEMBL5758142 0.85 GSK3B (0.72) GSK3BPRKACAPRKACGPRKACBPRKCG
SCHEMBL5759256 0.85 GSK3B (0.69) GSK3BPRKCGPRKCBPRKCAKCNH2
SCHEMBL9087475 0.79 PRKACA (0.82) GSK3BPRKACAPRKACGPRKACBPRKCG
SCHEMBL5754334 0.78 GSK3B (0.67) GSK3BPRKCGPRKCBPRKCAKCNH2
SCHEMBL5754325 0.77 GSK3B (0.69) GSK3BPRKCGPRKCBPRKCAKCNH2
SCHEMBL9085155 0.76 PRKACA (0.71) GSK3BPRKACAPRKACGPRKACBPRKCG
SCHEMBL9087381 0.76 PRKACA (0.82) GSK3BPRKACAPRKACGPRKACBPRKCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362047-B1 INDAZOLYL-SUBSTITUTED PYRROLINE COMPOUNDS AS KINASE INHIBITORS ORTHO MCNEIL PHARM INC (US) 2006-05-17 EP disclosed