SCHEMBL5758259

SCHEMBL5758259

OCCCc1ccc(SCc2coc(/C=C/c3ccccc3)n2)cc1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 11/20 0.39
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
HPGD P15428 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
KDM4E B2RXH2 1/20 0.37
LTB4R Q15722 3/20 0.36
MINK1 Q8N4C8 1/20 0.35
LTA4H P09960 1/20 0.33
EPHX2 P34913 1/20 0.33
CYP1A2 P05177 2/20 0.32
CYP2C19 P33261 2/20 0.32
CYP2D6 P10635 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP2C9 P11712 1/20 0.32
NPY1R P25929 1/20 0.32
NPY2R P49146 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5758262 1.00 ERBB2 (0.39) ERBB2MEN1KMT2AHPGDL3MBTL1
SCHEMBL5759912 0.85 FFAR1 (0.43) ERBB2MEN1KMT2AHPGDL3MBTL1
SCHEMBL5759910 0.85 FFAR1 (0.43) ERBB2MEN1KMT2AHPGDL3MBTL1
SCHEMBL5760787 0.81 LTB4R (0.37) ERBB2MEN1KMT2AHPGDL3MBTL1
SCHEMBL7959564 0.81 LTB4R (0.37) ERBB2MEN1KMT2AHPGDL3MBTL1
SCHEMBL5761322 0.81 ERBB2 (0.52) ERBB2MINK1LTA4HEPHX2
SCHEMBL5761318 0.81 ERBB2 (0.52) ERBB2MINK1LTA4HEPHX2
SCHEMBL5758381 0.81 CYP24A1 (0.43)
SCHEMBL5761435 0.81 CYP24A1 (0.43)
SCHEMBL5758992 0.80 CYP4F2 (0.42) KMT2AHPGDL3MBTL1KDM4ELTB4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1270571-B1 Heterocyclic compounds, their production and use TAKEDA PHARMACEUTICAL (JP) 2006-09-06 EP disclosed
EP-1270571-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-01-02 EP disclosed
US-6211215-B1 AROMATIC HETEROCYCLIC COMPOUND WITH AZOLE COMPOUND TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US disclosed