SCHEMBL5758402

SCHEMBL5758402

COC(=O)c1cc2cc(OCCC3CCCN3)ccc2o1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.47
CHEK2 O96017 1/20 0.44
ALDH1A1 P00352 3/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
MAOA P21397 1/20 0.43
TAS1R3 Q7RTX0 3/20 0.43
TAS1R1 Q7RTX1 3/20 0.43
KDM4E B2RXH2 3/20 0.42
MAPT P10636 2/20 0.42
HPGD P15428 2/20 0.42
HSD17B10 Q99714 2/20 0.42
AURKB Q96GD4 1/20 0.41
MKNK1 Q9BUB5 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4768815 0.88 PIM1 (0.48) MAOBCHEK2ALDH1A1MEN1KMT2A
SCHEMBL5760224 0.86 HPGD (0.48) MAOBCHEK2TAS1R3TAS1R1MAPT
SCHEMBL4764679 0.85 CHEK2 (0.49) MAOBCHEK2ALDH1A1MEN1KMT2A
SCHEMBL8902416 0.79 MAPT (0.57) CHEK2ALDH1A1MEN1KMT2AKDM4E
SCHEMBL445130 0.79 KDM4E (0.55) MAOBALDH1A1MAOAKDM4E
SCHEMBL9989067 0.79 MAOB (0.55) MAOBALDH1A1MEN1KMT2AMAOA
Hydrochloric Acid SCHEMBL5970288 0.77 CHEK2 (0.40) CHEK2TAS1R3TAS1R1HPGD
SCHEMBL6560708 0.76 MAPT (0.56) CHEK2ALDH1A1MEN1KMT2AKDM4E
SCHEMBL5105919 0.75 CYP1A2 (0.61) ALDH1A1MEN1KMT2AKDM4E
SCHEMBL6386675 0.74 XDH (0.52) MAOBALDH1A1KDM4EMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006042035-A2 METHOD OF MONITORING ANTI-TUMOR ACTIVITY OF AN HDAC INHIBITOR PHARMACYCLICS, INC. (US) 2006-04-20 WO disclosed
EP-1611088-A2 HYDROXAMATES AS THERAPEUTIC AGENTS AXYS PHARMACEUTICALS, INC. (US) 2006-01-04 EP disclosed
WO-2004092115-A2 HYDROXAMATES AS THERAPEUTIC AGENTS AXYS PHARMACEUTICALS INC. (US) 2004-10-28 WO disclosed