SCHEMBL5758990

SCHEMBL5758990

Cc1ccc(C(=O)N[C@@H](c2nc(=O)c(C)c(C)n2Cc2ccccc2)C(C)C)cc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.52
ALDH1A1 P00352 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
CYP3A4 P08684 2/20 0.51
CYP2C9 P11712 2/20 0.51
CYP2C19 P33261 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
KIF11 P52732 1/20 0.49
LMNA P02545 2/20 0.47
TP53 P04637 1/20 0.47
PPARG P37231 7/20 0.47
PKM P14618 1/20 0.41
FPR1 P21462 1/20 0.41
HDAC1 Q13547 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4359237 0.86 KIF11 (0.53) GAAALDH1A1SMN1; SMN2CYP3A4CYP2C9
SCHEMBL6454042 0.78 KIF11 (0.62) GAAALDH1A1CYP3A4CYP2C19KIF11
SCHEMBL1386243 0.76 LMNA (0.50) GAAALDH1A1SMN1; SMN2CYP3A4CYP2C9
SCHEMBL5752668 0.74 KIF11 (0.70) CYP3A4CYP2C19KIF11
SCHEMBL5758518 0.72 KIF11 (0.53) CYP3A4CYP2C19KIF11
SCHEMBL5755244 0.72 KIF11 (0.49) CYP3A4CYP2C19KIF11
SCHEMBL5756110 0.71 KIF11 (0.57) CYP3A4CYP2C19KIF11
SCHEMBL5754790 0.70 KIF11 (0.52) CYP3A4CYP2C19KIF11
SCHEMBL5863323 0.67 KIF11 (0.62) GAAKIF11TP53PPARGFPR1
SCHEMBL5754619 0.67 KIF11 (0.53) SMN1; SMN2CYP3A4CYP2C19KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1503993-A4 COMPOUNDS, METHODS AND COMPOSITIONS CYTOKINETICS INC (US) 2006-05-03 EP disclosed
EP-1503993-A2 COMPOUNDS, METHODS AND COMPOSITIONS Cytokinetics, Inc. (US) 2005-02-09 EP disclosed
WO-2003094839-A2 PYRIMIDINONE COMPOUNDS, COMPOSITIONS AND METHODS CYTOKINETICS, INC. (US) 2003-11-20 WO disclosed