SCHEMBL5761027

SCHEMBL5761027

ClCc1coc(-c2cccc(OCc3ccccc3)c2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 5/20 0.49
FFAR1 O14842 3/20 0.48
DRD2 P14416 1/20 0.45
DRD4 P21917 1/20 0.45
DRD3 P35462 1/20 0.45
PPARG P37231 3/20 0.44
MAOB P27338 3/20 0.43
BACE1 P56817 1/20 0.43
HPGD P15428 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
LMNA P02545 1/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ALDH1A1 P00352 1/20 0.43
XBP1 P17861 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5400326 0.86 FFAR1 (0.55) PPARAFFAR1DRD2DRD4DRD3
SCHEMBL4744758 0.85 PPARA (0.59) PPARAFFAR1DRD2DRD4DRD3
SCHEMBL3073429 0.83 FFAR1 (0.41) PPARAFFAR1DRD2DRD4DRD3
SCHEMBL4270619 0.82 KDM4E (0.49) FFAR1DRD2DRD4DRD3HPGD
SCHEMBL5186489 0.82 MAOB (0.49) PPARAMAOBHPGDNPC1RAB9A
SCHEMBL5015948 0.80 KDM4E (0.54) HPGDNPC1RAB9ALMNATSHR
SCHEMBL4896931 0.79 MRGPRX4 (0.53) PPARAMAOBALDH1A1
SCHEMBL4269852 0.79 KDM4E (0.53) DRD2DRD4DRD3HPGDNPC1
SCHEMBL4273714 0.78 KDM4E (0.50) HPGDNPC1RAB9ALMNATSHR
SCHEMBL1436020 0.78 DRD2 (0.58) PPARAFFAR1DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1270571-B1 Heterocyclic compounds, their production and use TAKEDA PHARMACEUTICAL (JP) 2006-09-06 EP disclosed
EP-1270571-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-01-02 EP disclosed
US-6211215-B1 AROMATIC HETEROCYCLIC COMPOUND WITH AZOLE COMPOUND TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US disclosed
EP-0912562-A1 HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1999-05-06 EP disclosed
WO-1998003505-A2 HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-01-29 WO disclosed