SCHEMBL5764241

SCHEMBL5764241

C#Cc1cc([Si](C)(C)C)cnc1N

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32
PTPN1 P18031 1/20 0.32
PTPN6 P29350 1/20 0.32
PTPN11 Q06124 1/20 0.32
P2RX3 P56373 2/20 0.31
P2RX2 Q9UBL9 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4877753 0.76 NOS3 (0.54) NOS3NOS1NOS2PTPN1PTPN6
SCHEMBL10017418 0.72 KMT2A (0.54) NOS3NOS1NOS2PTPN1PTPN6
SCHEMBL510587 0.72 PTPN1 (0.33) NOS3NOS1NOS2PTPN1PTPN6
SCHEMBL1748895 0.72 IDO1 (0.39) NOS3NOS1NOS2PTPN1PTPN6
SCHEMBL9538187 0.71 ACHE (0.32)
SCHEMBL1479446 0.70
SCHEMBL2060131 0.69 HTT (0.56) PTPN1PTPN6PTPN11
SCHEMBL6488816 0.67 MAP4K4 (0.44) NOS3NOS1NOS2
SCHEMBL8018559 0.67 EGFR (0.35)
SCHEMBL27827705 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114437037-B Compound containing pyridine-bis-triazole as well as preparation method and application thereof 西安交通大学 2023-04-07 CN claimed
CN-114437037-A Compound containing pyridine-bis-triazole as well as preparation method and application thereof 西安交通大学 2022-05-06 CN claimed
CN-114437037-B Compound containing pyridine-bis-triazole as well as preparation method and application thereof 西安交通大学 2023-04-07 CN disclosed
CN-114437037-A Compound containing pyridine-bis-triazole as well as preparation method and application thereof 西安交通大学 2022-05-06 CN disclosed
EP-1725544-A1 3-[4-HETEROCYCLYL-1,2,3-TRIAZOL-1-YL]-N-ARYL-BENZAMIDES AS INHIBITORS OF THE CYTOKINES PRODUCTION FOR THE TREATMENT OF CHRONIC INFLAMMATORY DISEASES BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2006-11-29 EP disclosed
WO-2005090333-A1 3-‘4-HETEROCYCLYL -1,2,3,-TRIAZOL-1-YL!-N-ARYL-BENZAMIDES AS INHIBITORS OF THE CYTOKINES PRODUCTION FOR THE TREATMENT OF CHRONIC INFLAMMATORY DISEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-09-29 WO disclosed