SCHEMBL5764950

SCHEMBL5764950

COc1ccc2nccc(NC(=O)OC3CCN(CCc4ccc5c(c4)NC(=O)CO5)CC3)c2n1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 13/20 0.51
HTR1D P28221 9/20 0.51
HTR1B P28222 7/20 0.51
SLC6A4 P31645 6/20 0.47
KCNH2 Q12809 6/20 0.47
DRD2 P14416 2/20 0.44
HTR2A P28223 2/20 0.44
HTR2B P41595 2/20 0.44
ADRB1 P08588 1/20 0.44
HTR7 P34969 1/20 0.44
DRD3 P35462 1/20 0.44
HTR2C P28335 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14573146 0.90 KCNH2 (0.49) HTR1AHTR1DHTR1BSLC6A4KCNH2
SCHEMBL5764977 0.88 HTR1D (0.53) HTR1AHTR1DHTR1BKCNH2
SCHEMBL5765233 0.86 SLC2A1 (0.43) HTR1AHTR1DKCNH2
SCHEMBL5764668 0.86 KCNH2 (0.53) KCNH2
SCHEMBL5764517 0.86 KCNH2 (0.58) KCNH2
SCHEMBL5764669 0.86 KCNH2 (0.45) KCNH2
SCHEMBL5764847 0.83 KCNH2 (0.48) KCNH2
SCHEMBL5765881 0.83 KCNH2 (0.45) KCNH2
SCHEMBL5763984 0.82 KCNH2 (0.45) HTR1ASLC6A4KCNH2
SCHEMBL6684945 0.79 HTR1A (0.40) HTR1AHTR1DHTR1BSLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392686-B1 BICYCLIC NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVES FOR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2006-10-18 EP claimed