SCHEMBL5765604

SCHEMBL5765604

CS(=O)(=O)OCC1CCN(Cc2ccccc2)C1.OC1CCN(Cc2ccccc2)C1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.53
DRD2 P14416 3/20 0.49
DRD4 P21917 3/20 0.49
SPHK1 Q9NYA1 2/20 0.47
SPHK2 Q9NRA0 1/20 0.47
BCHE P06276 4/20 0.47
ACHE P22303 4/20 0.47
MAOB P27338 2/20 0.46
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
DRD3 P35462 2/20 0.44
CCR3 P51677 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4917475 0.93 DRD2 (0.52) ALDH1A1DRD2DRD4BCHEACHE
SCHEMBL2576650 0.93 DRD2 (0.52) ALDH1A1DRD2DRD4BCHEACHE
SCHEMBL4917481 0.93 DRD2 (0.52) ALDH1A1DRD2DRD4BCHEACHE
SCHEMBL2454072 0.85 BCHE (0.58) ALDH1A1BCHEACHEMAOB
SCHEMBL12090230 0.85 BCHE (0.58) ALDH1A1BCHEACHEMAOB
SCHEMBL5743125 0.84 ALDH1A1 (0.66) ALDH1A1DRD2SPHK1SPHK2BCHE
SCHEMBL5744592 0.84 ALDH1A1 (0.66) ALDH1A1DRD2SPHK1SPHK2BCHE
SCHEMBL6279418 0.82 ALDH1A1 (0.57) ALDH1A1SPHK1SPHK2BCHEACHE
SCHEMBL9217317 0.80 HTR2A (0.55) ALDH1A1DRD2DRD4BCHEACHE
SCHEMBL608225 0.79 ALDH1A1 (0.81) ALDH1A1BCHEACHENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1474135-A4 INDOLE, AZAINDOLE AND RELATED HETEROCYCLIC PYRROLIDINE DERIVATIVES BRISTOL MYERS SQUIBB CO (US) 2006-01-18 EP disclosed
EP-1474135-A1 INDOLE, AZAINDOLE AND RELATED HETEROCYCLIC PYRROLIDINE DERIVATIVES Bristol-Myers Squibb Company (US) 2004-11-10 EP disclosed
WO-2003068221-A1 INDOLE, AZAINDOLE AND RELATED HETEROCYCLIC PYRROLIDINE DERIVATIVES BRISTOL-MYERS SQUIBB COMPANY (US) 2003-08-21 WO disclosed