SCHEMBL5767040

SCHEMBL5767040

COc1cc2sc(C(=O)Nc3nnn[nH]3)c(SCC3CC3)c2cc1OC

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.39
STING1 Q86WV6 1/20 0.34
METAP2 P50579 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
PDE4B Q07343 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
ABCC8 Q09428 2/20 0.31
KCNJ11 Q14654 2/20 0.31
ESR1 P03372 1/20 0.31
ALPL P05186 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6808614 0.82 POLB (0.40) STING1NPC1RAB9AMEN1KMT2A
SCHEMBL6817003 0.80 EDNRA (0.41) PIK3CDSTING1L3MBTL1ESR1MEN1
SCHEMBL6812458 0.79 L3MBTL1 (0.38) L3MBTL1ALPLMEN1KMT2A
SCHEMBL6808610 0.79 STING1 (0.51) STING1NPC1RAB9AMEN1KMT2A
SCHEMBL6808644 0.79 PDGFRA (0.35) PIK3CDSTING1L3MBTL1ESR1ALPL
SCHEMBL6812307 0.78 KMT2A (0.39) STING1NPC1RAB9AMEN1KMT2A
SCHEMBL4790749 0.78 L3MBTL1 (0.37) NPC1RAB9AL3MBTL1ESR1MEN1
SCHEMBL6812764 0.78 AURKB (0.33) PIK3CDSTING1NPC1RAB9AL3MBTL1
SCHEMBL6811963 0.78 KDM4E (0.39) PIK3CDSTING1NPC1RAB9AL3MBTL1
SCHEMBL6812848 0.78 EDNRA (0.47) L3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636212-A1 CYCLOALKYLSULFANYL SUBSTITUTED BENZO[B]THIOPHENES AS THERAPEUTIC AGENTS Warner-Lambert Company LLC (US) 2006-03-22 EP disclosed
WO-2004108714-A1 CYCLOALKYLSULFANYL SUBSTITUTED BENZO[B]THIOPHENES AS THERAPEUTIC AGENTS WARNER-LAMBERT COMPANY LLC (US) 2004-12-16 WO disclosed