SCHEMBL5768428

SCHEMBL5768428

COC(=O)C(=O)c1cn2c3c(cccc13)CCN(C(=O)OC(C)(C)C)CC2

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.40
ESR2 Q92731 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39
NAMPT P43490 1/20 0.39
NR1H2 P55055 1/20 0.39
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
GBA1 P04062 2/20 0.38
POLB P06746 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LIPG Q9Y5X9 1/20 0.37
DTYMK P23919 1/20 0.37
STS P08842 1/20 0.37
THRB P10828 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1719811 0.80 MTNR1A (0.51) ALDH1A1
SCHEMBL5768646 0.79 MTNR1A (0.47) ALDH1A1
SCHEMBL3050216 0.78 LIPG (0.51) ESR2CHRM2CHRM4CHRM1CHRM3
SCHEMBL20434858 0.77 ESR2 (0.39) ESR2NAMPTNR1H2LMNATP53
SCHEMBL13056761 0.76 PARP1 (0.41) ALDH1A1
SCHEMBL21577586 0.75 MAPT (0.41) ESR2NAMPTNR1H2ALDH1A1LIPG
SCHEMBL8363597 0.75 NAMPT (0.38) NAMPTNR1H2LMNATP53POLB
SCHEMBL2018775 0.75 POLB (0.51) LMNAPOLBTHRB
SCHEMBL2261638 0.74 ESR2 (0.45) ESR2NAMPTNR1H2LMNATP53
SCHEMBL10234454 0.73 TMEM97 (0.44) LIPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1483265-B1 PURINE DERIVATIVES AS KINASE INHIBITORS LILLY CO ELI (US) 2006-11-22 EP disclosed