SCHEMBL5769191

SCHEMBL5769191

CNCc1cnccc1Cl

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 8/20 0.55
SLC6A4 P31645 8/20 0.55
CYP2A6 P11509 2/20 0.41
SLC6A3 Q01959 2/20 0.40
AOC1 P19801 2/20 0.39
AOC3 Q16853 2/20 0.39
MAPK8 P45983 1/20 0.39
PRMT6 Q96LA8 2/20 0.38
EPHX2 P34913 1/20 0.38
GAA P10253 1/20 0.38
TAAR1 Q96RJ0 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
PRKCI P41743 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5768459 0.84 SLC6A2 (0.51) SLC6A2SLC6A4CYP2A6SLC6A3AOC1
SCHEMBL25910954 0.83 CYP1A2 (0.42) SLC6A2SLC6A4GAACYP2D6CYP2C19
Hydrochloric Acid SCHEMBL31407242 0.82 SLC6A2 (0.50) SLC6A2SLC6A4CYP2A6SLC6A3AOC1
SCHEMBL10268296 0.77
SCHEMBL31651986 0.77
SCHEMBL25378025 0.76 SLC6A2 (0.44) SLC6A2SLC6A4CYP2A6AOC1AOC3
SCHEMBL12836473 0.76 SLC6A2 (0.54) SLC6A2SLC6A4CYP2A6SLC6A3AOC1
SCHEMBL13456619 0.76 SLC6A2 (0.44) SLC6A2SLC6A4CYP2A6AOC1AOC3
SCHEMBL16547439 0.76 SLC6A2 (0.54) SLC6A2SLC6A4CYP2A6SLC6A3AOC1
Hydrochloric Acid SCHEMBL11467876 0.75 CYP2E1 (0.43) SLC6A2SLC6A4CYP2A6SLC6A3AOC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120165351-A1 QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2012-06-28 US disclosed
US-20060160794-A1 Tachykinin receptor antagonists ELI LILLY AND COMPANY 2006-07-20 US disclosed
EP-1638944-A1 TACHYKININ RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2006-03-29 EP disclosed
WO-2005000821-A1 TACHYKININ RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2005-01-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060160794-A1 Tachykinin receptor antagonists TACR1, TACR2, PROKR1 SLC6A2 221/4885SLC6A4 348/4885CYP2A6 3531/4885
US-20120165351-A1 QUINAZOLINE DERIVATIVES AQP1, F12, AQP3 SLC6A2 756/4885SLC6A4 679/4885CYP2A6 2387/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.